Assay Detail
Functional
CHEMBL3720724
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Inhibition of cell proliferation of human Jurkat cells incubated for 72 hrs by Alamar blue assay
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Jurkat |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Family of PFKFB3 inhibitors with anti-neoplastic activities
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 25 | 5.55 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3716423 | — | — | 1 | 6.22 |
| CHEMBL3718583 | — | — | 1 | 6.22 |
| CHEMBL3715765 | — | — | 1 | 6.05 |
| CHEMBL3718122 | — | — | 1 | 6.05 |
| CHEMBL3718476 | — | — | 1 | 6.00 |
| CHEMBL3717731 | — | — | 1 | 6.00 |
| CHEMBL3718751 | — | — | 1 | 6.00 |
| CHEMBL3715519 | — | — | 1 | 5.89 |
| CHEMBL3719281 | — | — | 1 | 5.77 |
| CHEMBL3717996 | — | — | 1 | 5.62 |
| CHEMBL3715718 | — | — | 1 | 5.60 |
| CHEMBL3717919 | — | — | 1 | 5.60 |
| CHEMBL3718600 | — | — | 1 | 5.60 |
| CHEMBL3715613 | — | — | 1 | 5.51 |
| CHEMBL3717367 | — | — | 1 | 5.43 |
| CHEMBL3717735 | — | — | 1 | 5.38 |
| CHEMBL3715989 | — | — | 1 | 5.32 |
| CHEMBL3714967 | — | — | 1 | 5.31 |
| CHEMBL3716040 | — | — | 1 | 5.26 |
| CHEMBL3718103 | — | — | 1 | 5.19 |
| CHEMBL3716953 | — | — | 1 | 4.85 |
| CHEMBL3717112 | — | — | 1 | 4.77 |
| CHEMBL3401545 | — | — | 1 | 4.09 |
| CHEMBL3715996 | — | — | 1 | - |
| CHEMBL3715205 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3716423 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3718583 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL3715765 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL3718122 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL3718476 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL3717731 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL3718751 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL3715519 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL3719281 | — | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL3717996 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL3715718 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL3717919 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL3718600 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL3715613 | — | IC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL3717367 | — | IC50 | = | 3700.0 | nM | 5.43 |
| CHEMBL3717735 | — | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL3715989 | — | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL3714967 | — | IC50 | = | 4900.0 | nM | 5.31 |
| CHEMBL3716040 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL3718103 | — | IC50 | = | 6400.0 | nM | 5.19 |
| CHEMBL3716953 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL3717112 | — | IC50 | = | 17000.0 | nM | 4.77 |
| CHEMBL3401545 | — | IC50 | = | 80500.0 | nM | 4.09 |
| CHEMBL3715996 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL3715205 | — | IC50 | > | 4000.0 | nM | - |