Assay Detail
Functional
CHEMBL3757808
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Antiproliferative activity against human DLD1 cells after 72 hrs by MTT assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | DLD-1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis and biological evaluation of novel 7-O-lipophilic substituted baicalein derivatives as potential anticancer agents
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.19 | 5.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3753264 | — | — | 1 | 5.21 |
| CHEMBL3754716 | — | — | 1 | 5.16 |
| CHEMBL8260 | BAICALEIN | 2.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3753264 | — | IC50 | = | 6190.0 | nM | 5.21 |
| CHEMBL3754716 | — | IC50 | = | 6860.0 | nM | 5.16 |
| CHEMBL8260 | BAICALEIN | IC50 | > | 20000.0 | nM | - |