Assay Detail
Functional
CHEMBL3760689
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Partial agonist activity at human mu opioid receptor expressed in CHO cells by [35S]GTPgammaS binding
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Multitarget opioid ligands in pain relief: New players in an old game.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Emax | 1 | - | - |
| EC50 | 1 | 8.89 | 8.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL147511 | — | — | 1 | 8.89 |
| CHEMBL146756 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL147511 | — | EC50 | = | 1.3 | nM | 8.89 |
| CHEMBL146756 | — | Emax | = | 42.0 | % | - |