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Assay Detail

CHEMBL3762579

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]DSLET from delta opioid receptor in rat brain membrane
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Tissue Brain
Subcellular Membrane
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Delta-type opioid receptor (CHEMBL269)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Multitarget opioid ligands in pain relief: New players in an old game.
Turnaturi R, Aricò G, Ronsisvalle G, Parenti C, Pasquinucci L.
Eur J Med Chem (2016) 108 : 211 -228
PubMed 26656913 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.52 8.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL557035 1 8.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL557035 Ki = 3.0 nM 8.52