Assay Detail
Functional
CHEMBL3854071
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Antiviral activity against Influenza A virus A/PR/8/34 (H1N1) infected in MDCK cells assessed as reduction in plaque formation after 2 days by plaque reduction assay
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Influenza A virus (A/Puerto Rico/8/1934(H1N1)) |
| Cell Type | MDCK |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Polymerase Acidic Protein-Basic Protein 1 (PA-PB1) Protein-Protein Interaction as a Target for Next-Generation Anti-influenza Therapeutics.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 9 | 4.72 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3577824 | — | — | 1 | 6.00 |
| CHEMBL3947563 | — | — | 1 | 5.00 |
| CHEMBL3288047 | — | — | 1 | 4.73 |
| CHEMBL284733 | DICLAZURIL | 2.0 | 1 | 4.51 |
| CHEMBL388590 | BENZBROMARONE | 4.0 | 1 | 4.41 |
| CHEMBL1698011 | TRENBOLONE ACETATE | 2.0 | 1 | 4.29 |
| CHEMBL3288048 | — | — | 1 | 4.12 |
| CHEMBL3945111 | — | — | 1 | - |
| CHEMBL3577796 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3577824 | — | EC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL3947563 | — | EC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL3288047 | — | EC50 | = | 18600.0 | nM | 4.73 |
| CHEMBL284733 | DICLAZURIL | EC50 | = | 31000.0 | nM | 4.51 |
| CHEMBL388590 | BENZBROMARONE | EC50 | = | 39000.0 | nM | 4.41 |
| CHEMBL1698011 | TRENBOLONE ACETATE | EC50 | = | 51000.0 | nM | 4.29 |
| CHEMBL3288048 | — | EC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL3945111 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL3577796 | — | EC50 | > | 100000.0 | nM | - |