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Assay Detail

CHEMBL3856719

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Protection against t-BHP-induced oxidative injury in rat H9c2 cells assessed as increase in cell viability incubated for 10 mins followed by stimulation with t-BHP for 24 hrs by neutral red staining based assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Rattus norvegicus
Cell Type H9c2
Confidence 1 — Organism
Curated By Autocuration

Target

H9c2 (CHEMBL614576)
Type CELL-LINE
Organism Rattus norvegicus

Publication

Aroylhydrazone iron chelators: Tuning antioxidant and antiproliferative properties by hydrazide modifications.
Hrušková K, Potůčková E, Hergeselová T, Liptáková L, Hašková P, Mingas P, Kovaříková P, Šimůnek T, Vávrová K.
Eur J Med Chem (2016) 120 : 97 -110
PubMed 27187862 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 4.81 4.94

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2261891 1 4.94
CHEMBL3975887 1 4.75
CHEMBL201761 SALINAZID 2.0 1 4.74

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2261891 EC50 = 11400.0 nM 4.94
CHEMBL3975887 EC50 = 17800.0 nM 4.75
CHEMBL201761 SALINAZID EC50 = 18200.0 nM 4.74