Assay Detail
Functional
CHEMBL3862205
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Cytotoxicity against human PC3 cells assessed as decrease in cell viability after 72 hrs by MTT assay
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | PC-3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 5.56 | 6.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3983705 | — | — | 1 | 6.39 |
| CHEMBL3963286 | — | — | 1 | 5.89 |
| CHEMBL3916732 | — | — | 1 | 5.87 |
| CHEMBL3980519 | — | — | 1 | 5.68 |
| CHEMBL3936130 | — | — | 1 | 5.66 |
| CHEMBL3945406 | — | — | 1 | 5.59 |
| CHEMBL3986488 | — | — | 1 | 5.56 |
| CHEMBL3911886 | — | — | 1 | 5.51 |
| CHEMBL3974809 | — | — | 1 | 5.47 |
| CHEMBL3952951 | — | — | 1 | 5.36 |
| CHEMBL3973814 | — | — | 1 | 5.24 |
| CHEMBL3901778 | — | — | 1 | 5.16 |
| CHEMBL3908949 | — | — | 1 | 4.91 |
| CHEMBL3927420 | — | — | 1 | - |
| CHEMBL3941393 | — | — | 1 | - |
| CHEMBL3970985 | — | — | 1 | - |
| CHEMBL3965105 | — | — | 1 | - |
| CHEMBL1098852 | — | — | 1 | - |
| CHEMBL3944199 | — | — | 1 | - |
| CHEMBL3916262 | — | — | 1 | - |
| CHEMBL3935226 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3983705 | — | IC50 | = | 410.0 | nM | 6.39 |
| CHEMBL3963286 | — | IC50 | = | 1290.0 | nM | 5.89 |
| CHEMBL3916732 | — | IC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL3980519 | — | IC50 | = | 2070.0 | nM | 5.68 |
| CHEMBL3936130 | — | IC50 | = | 2170.0 | nM | 5.66 |
| CHEMBL3945406 | — | IC50 | = | 2550.0 | nM | 5.59 |
| CHEMBL3986488 | — | IC50 | = | 2770.0 | nM | 5.56 |
| CHEMBL3911886 | — | IC50 | = | 3070.0 | nM | 5.51 |
| CHEMBL3974809 | — | IC50 | = | 3420.0 | nM | 5.47 |
| CHEMBL3952951 | — | IC50 | = | 4370.0 | nM | 5.36 |
| CHEMBL3973814 | — | IC50 | = | 5730.0 | nM | 5.24 |
| CHEMBL3901778 | — | IC50 | = | 6910.0 | nM | 5.16 |
| CHEMBL3908949 | — | IC50 | = | 12440.0 | nM | 4.91 |
| CHEMBL3927420 | — | IC50 | > | 12980.0 | nM | - |
| CHEMBL3941393 | — | IC50 | > | 9780.0 | nM | - |
| CHEMBL3970985 | — | IC50 | > | 12980.0 | nM | - |
| CHEMBL3965105 | — | IC50 | > | 8480.0 | nM | - |
| CHEMBL1098852 | — | IC50 | - | — | - | |
| CHEMBL3944199 | — | IC50 | > | 14000.0 | nM | - |
| CHEMBL3916262 | — | IC50 | > | 14000.0 | nM | - |
| CHEMBL3935226 | — | IC50 | > | 10350.0 | nM | - |