Assay Detail
Binding
CHEMBL3882380
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of rat liver CK2 using RRADDSDDDDD as substrate after 10 mins in presence of [gamma-33P]-ATP
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Use of dibenzofuranone derivatives to inhibit kinases
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.79 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3974619 | — | — | 1 | 7.00 |
| CHEMBL29898 | QUINALIZARIN | — | 1 | 6.96 |
| CHEMBL3911092 | — | — | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3974619 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL29898 | QUINALIZARIN | IC50 | = | 110.0 | nM | 6.96 |
| CHEMBL3911092 | — | IC50 | = | 400.0 | nM | 6.40 |