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Assay Detail

CHEMBL4004666

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of CYP2C9 in human liver microsomes using tolbutamide as substrate after 5 to 15 mins
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Tissue Liver
Subcellular Microsomes
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 2C9 (CHEMBL3397)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of GBT440, an Orally Bioavailable R-State Stabilizer of Sickle Cell Hemoglobin.
Metcalf B, Chuang C, Dufu K, Patel MP, Silva-Garcia A, Johnson C, Lu Q, Partridge JR, Patskovska L, Patskovsky Y, Almo SC, Jacobson MP, Hua L, Xu Q, Gwaltney SL, Yee C, Harris J, Morgan BP, James J, Xu D, Hutchaleelaha A, Paulvannan K, Oksenberg D, Li Z.
ACS Med Chem Lett (2017) 8 : 321 -326
PubMed 28337324 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.88 6.69

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1109 SULFAPHENAZOLE 4.0 1 6.69
CHEMBL4101807 VOXELOTOR 4.0 1 5.07

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1109 SULFAPHENAZOLE IC50 = 205.0 nM 6.69
CHEMBL4101807 VOXELOTOR IC50 = 8500.0 nM 5.07