Assay Detail
ADMET
CHEMBL4013734
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at mouse NMUR1 expressed in CHO cells assessed as induction of Ca2+ flux measured for 180 secs by Fluo 4-AM dye-based FLIPR assay
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Potent Body Weight-Lowering Effect of a Neuromedin U Receptor 2-selective PEGylated Peptide.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 27 | 8.36 | 9.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4088263 | — | — | 1 | 9.80 |
| CHEMBL4068681 | — | — | 1 | 9.68 |
| CHEMBL4095998 | — | — | 1 | 9.57 |
| CHEMBL4098010 | — | — | 1 | 9.24 |
| CHEMBL3356083 | — | — | 1 | 9.23 |
| CHEMBL4073946 | — | — | 1 | 9.16 |
| CHEMBL4099780 | — | — | 1 | 8.60 |
| CHEMBL4059530 | — | — | 1 | 8.52 |
| CHEMBL4079986 | — | — | 1 | 8.47 |
| CHEMBL4063830 | — | — | 1 | 8.43 |
| CHEMBL4081760 | — | — | 1 | 8.26 |
| CHEMBL4061507 | — | — | 1 | 8.24 |
| CHEMBL4089636 | — | — | 1 | 8.13 |
| CHEMBL4090300 | — | — | 1 | 8.10 |
| CHEMBL4091611 | — | — | 1 | 8.07 |
| CHEMBL4063341 | — | — | 1 | 8.02 |
| CHEMBL4087867 | — | — | 1 | 7.89 |
| CHEMBL4100718 | — | — | 1 | 7.64 |
| CHEMBL4097355 | — | — | 1 | 7.55 |
| CHEMBL4060571 | — | — | 1 | 7.42 |
| CHEMBL4082455 | — | — | 1 | 7.08 |
| CHEMBL4092033 | — | — | 1 | 6.80 |
| CHEMBL4060027 | — | — | 1 | - |
| CHEMBL4071218 | — | — | 1 | - |
| CHEMBL4070175 | — | — | 1 | - |
| CHEMBL4091208 | — | — | 1 | - |
| CHEMBL4069256 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4088263 | — | EC50 | = | 0.16 | nM | 9.80 |
| CHEMBL4068681 | — | EC50 | = | 0.21 | nM | 9.68 |
| CHEMBL4095998 | — | EC50 | = | 0.27 | nM | 9.57 |
| CHEMBL4098010 | — | EC50 | = | 0.57 | nM | 9.24 |
| CHEMBL3356083 | — | EC50 | = | 0.59 | nM | 9.23 |
| CHEMBL4073946 | — | EC50 | = | 0.69 | nM | 9.16 |
| CHEMBL4099780 | — | EC50 | = | 2.5 | nM | 8.60 |
| CHEMBL4059530 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL4079986 | — | EC50 | = | 3.4 | nM | 8.47 |
| CHEMBL4063830 | — | EC50 | = | 3.7 | nM | 8.43 |
| CHEMBL4081760 | — | EC50 | = | 5.5 | nM | 8.26 |
| CHEMBL4061507 | — | EC50 | = | 5.8 | nM | 8.24 |
| CHEMBL4089636 | — | EC50 | = | 7.4 | nM | 8.13 |
| CHEMBL4090300 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL4091611 | — | EC50 | = | 8.5 | nM | 8.07 |
| CHEMBL4063341 | — | EC50 | = | 9.6 | nM | 8.02 |
| CHEMBL4087867 | — | EC50 | = | 13.0 | nM | 7.89 |
| CHEMBL4100718 | — | EC50 | = | 23.0 | nM | 7.64 |
| CHEMBL4097355 | — | EC50 | = | 28.0 | nM | 7.55 |
| CHEMBL4060571 | — | EC50 | = | 38.0 | nM | 7.42 |
| CHEMBL4082455 | — | EC50 | = | 83.0 | nM | 7.08 |
| CHEMBL4092033 | — | EC50 | = | 160.0 | nM | 6.80 |
| CHEMBL4060027 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4071218 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4070175 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4091208 | — | EC50 | > | 1000.0 | nM | - |
| CHEMBL4069256 | — | EC50 | > | 1000.0 | nM | - |