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Assay Detail

CHEMBL4133995

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Chikungunya virus Indian ocean strain 899 infected in African green monkey Vero cells assessed as reduction in virus-induced cytopathic effect by MTS assay
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Chikungunya virus
Cell Type Vero
Confidence 1 — Organism
Curated By Intermediate

Target

Chikungunya virus (CHEMBL4296563)
Type ORGANISM
Organism Chikungunya virus

Publication

Environmentally Friendly Procedure Based on Supercritical Fluid Chromatography and Tandem Mass Spectrometry Molecular Networking for the Discovery of Potent Antiviral Compounds from Euphorbia semiperfoliata.
Nothias LF, Boutet-Mercey S, Cachet X, De La Torre E, Laboureur L, Gallard JF, Retailleau P, Brunelle A, Dorrestein PC, Costa J, Bedoya LM, Roussi F, Leyssen P, Alcami J, Paolini J, Litaudon M, Touboul D.
J Nat Prod (2017) 80 : 2620 -2629
PubMed 28925702 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 8 5.77 8.54

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL279115 PHORBOL MYRISTATE ACETATE 2.0 1 8.54
CHEMBL4170130 1 6.36
CHEMBL4165007 1 6.00
CHEMBL170518 PROSTRATIN 1 5.58
CHEMBL4169508 1 4.86
CHEMBL2375779 1 4.77
CHEMBL4168419 1 4.29
CHEMBL4174527 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL279115 PHORBOL MYRISTATE ACETATE EC50 = 2.9 nM 8.54
CHEMBL4170130 EC50 = 440.0 nM 6.36
CHEMBL4165007 EC50 = 1000.0 nM 6.00
CHEMBL170518 PROSTRATIN EC50 = 2600.0 nM 5.58
CHEMBL4169508 EC50 = 13800.0 nM 4.86
CHEMBL2375779 EC50 = 17000.0 nM 4.77
CHEMBL4168419 EC50 = 51100.0 nM 4.29
CHEMBL4174527 EC50 > 153000.0 nM -