Assay Detail
Functional
CHEMBL4135029
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against Human respiratory syncytial virus A2 ATCC VR 1540 infected in African green monkey Vero 76 cells assessed as protection against virus-induced cytopathic effect after 5 days by crystal violet staining-based plaque reduction assay
32
Total Activities
32
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Human respiratory syncytial virus A2 |
| Cell Type | Vero 76 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Inhibitors of Yellow Fever Virus replication based on 1,3,5-triphenyl-4,5-dihydropyrazole scaffold: Design, synthesis and antiviral evaluation.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 32 | 5.16 | 5.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1643 | RIBAVIRIN | 4.0 | 1 | 5.92 |
| CHEMBL564201 | 6-AZAURIDINE | — | 1 | 4.40 |
| CHEMBL1441897 | — | — | 1 | - |
| CHEMBL1514645 | — | — | 1 | - |
| CHEMBL1591211 | — | — | 1 | - |
| CHEMBL4166223 | — | — | 1 | - |
| CHEMBL4168561 | — | — | 1 | - |
| CHEMBL1867917 | — | — | 1 | - |
| CHEMBL1881501 | — | — | 1 | - |
| CHEMBL4173042 | — | — | 1 | - |
| CHEMBL4166621 | — | — | 1 | - |
| CHEMBL4174536 | — | — | 1 | - |
| CHEMBL4159714 | — | — | 1 | - |
| CHEMBL4170341 | — | — | 1 | - |
| CHEMBL4163087 | — | — | 1 | - |
| CHEMBL1565276 | — | — | 1 | - |
| CHEMBL4166525 | — | — | 1 | - |
| CHEMBL4177143 | — | — | 1 | - |
| CHEMBL4169949 | — | — | 1 | - |
| CHEMBL4162022 | — | — | 1 | - |
| CHEMBL4164614 | — | — | 1 | - |
| CHEMBL4175245 | — | — | 1 | - |
| CHEMBL4176360 | — | — | 1 | - |
| CHEMBL4165746 | — | — | 1 | - |
| CHEMBL4161254 | — | — | 1 | - |
| CHEMBL4169180 | — | — | 1 | - |
| CHEMBL4169590 | — | — | 1 | - |
| CHEMBL4177444 | — | — | 1 | - |
| CHEMBL4172978 | — | — | 1 | - |
| CHEMBL4173795 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1643 | RIBAVIRIN | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL564201 | 6-AZAURIDINE | EC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL4163087 | — | EC50 | > | 88000.0 | nM | - |
| CHEMBL4169900 | — | EC50 | > | 28000.0 | nM | - |
| CHEMBL4170341 | — | EC50 | > | 29000.0 | nM | - |
| CHEMBL4159714 | — | EC50 | > | 25000.0 | nM | - |
| CHEMBL4174536 | — | EC50 | > | 28000.0 | nM | - |
| CHEMBL4166621 | — | EC50 | > | 96000.0 | nM | - |
| CHEMBL4173042 | — | EC50 | > | 35000.0 | nM | - |
| CHEMBL1881501 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL1867917 | — | EC50 | > | 25000.0 | nM | - |
| CHEMBL4168561 | — | EC50 | > | 24000.0 | nM | - |
| CHEMBL4166223 | — | EC50 | > | 21000.0 | nM | - |
| CHEMBL1591211 | — | EC50 | > | 21000.0 | nM | - |
| CHEMBL1514645 | — | EC50 | > | 26000.0 | nM | - |
| CHEMBL1441897 | — | EC50 | > | 23000.0 | nM | - |
| CHEMBL1530025 | — | EC50 | > | 24000.0 | nM | - |
| CHEMBL1565276 | — | EC50 | > | 22000.0 | nM | - |
| CHEMBL4166525 | — | EC50 | > | 14000.0 | nM | - |
| CHEMBL4177143 | — | EC50 | > | 14000.0 | nM | - |
| CHEMBL4169949 | — | EC50 | > | 20000.0 | nM | - |
| CHEMBL4162022 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4164614 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4175245 | — | EC50 | > | 25000.0 | nM | - |
| CHEMBL4176360 | — | EC50 | > | 90000.0 | nM | - |
| CHEMBL4165746 | — | EC50 | > | 92000.0 | nM | - |
| CHEMBL4161254 | — | EC50 | > | 85000.0 | nM | - |
| CHEMBL4169180 | — | EC50 | > | 82000.0 | nM | - |
| CHEMBL4169590 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4177444 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4172978 | — | EC50 | > | 100000.0 | nM | - |
| CHEMBL4173795 | — | EC50 | > | 88000.0 | nM | - |