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Assay Detail

CHEMBL4146837

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of equine serum BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition measured every minute for 10 mins by Ellman's method
61
Total Activities
57
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Equus caballus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cholinesterase (CHEMBL5763)
Type SINGLE PROTEIN
Organism Equus caballus

Publication

Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine "bio-oxidizable" prodrugs: Synthesis, biological evaluation and structure-activity relationship.
Azzouz R, Peauger L, Gembus V, Ţînţaş ML, Sopková-de Oliveira Santos J, Papamicaël C, Levacher V.
Eur J Med Chem (2018) 145 : 165 -190
PubMed 29324339 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 61 5.73 8.49

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL95 TACRINE 4.0 1 8.49
CHEMBL4177133 1 6.59
CHEMBL4176179 1 6.47
CHEMBL4159243 1 6.43
CHEMBL4160115 1 6.38
CHEMBL4161065 1 6.36
CHEMBL4168037 1 6.31
CHEMBL4166513 1 6.30
CHEMBL4168987 1 6.22
CHEMBL4173239 1 6.18
CHEMBL4160696 4 5.78
CHEMBL4165327 1 5.75
CHEMBL4171568 1 5.69
CHEMBL4173405 1 5.66
CHEMBL4164981 1 5.65
CHEMBL4170530 1 5.60
CHEMBL4166464 1 5.58
CHEMBL4165562 1 5.50
CHEMBL4162993 1 5.49
CHEMBL502 DONEPEZIL 4.0 1 5.47
CHEMBL4170614 1 5.40
CHEMBL4172797 1 5.38
CHEMBL4173784 1 5.38
CHEMBL4159880 1 5.37
CHEMBL4174056 1 5.36
CHEMBL4169887 1 5.27
CHEMBL4162692 1 5.24
CHEMBL4166141 1 5.22
CHEMBL4172353 1 5.21
CHEMBL4174372 1 5.04

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL95 TACRINE IC50 = 3.2 nM 8.49
CHEMBL4177133 IC50 = 256.0 nM 6.59
CHEMBL4176179 IC50 = 341.0 nM 6.47
CHEMBL4159243 IC50 = 373.2 nM 6.43
CHEMBL4160115 IC50 = 412.0 nM 6.38
CHEMBL4161065 IC50 = 433.0 nM 6.36
CHEMBL4168037 IC50 = 489.0 nM 6.31
CHEMBL4166513 IC50 = 496.0 nM 6.30
CHEMBL4168987 IC50 = 596.0 nM 6.22
CHEMBL4173239 IC50 = 665.0 nM 6.18
CHEMBL4160696 IC50 = 1670.0 nM 5.78
CHEMBL4165327 IC50 = 1790.0 nM 5.75
CHEMBL4160696 IC50 = 1830.0 nM 5.74
CHEMBL4171568 IC50 = 2035.0 nM 5.69
CHEMBL4173405 IC50 = 2170.0 nM 5.66
CHEMBL4164981 IC50 = 2239.0 nM 5.65
CHEMBL4170530 IC50 = 2505.0 nM 5.60
CHEMBL4166464 IC50 = 2637.1 nM 5.58
CHEMBL4165562 IC50 = 3198.0 nM 5.50
CHEMBL4162993 IC50 = 3264.0 nM 5.49
CHEMBL502 DONEPEZIL IC50 = 3365.0 nM 5.47
CHEMBL4170614 IC50 = 4020.0 nM 5.40
CHEMBL4160696 IC50 = 3970.0 nM 5.40
CHEMBL4173784 IC50 = 4147.0 nM 5.38
CHEMBL4172797 IC50 = 4140.0 nM 5.38
CHEMBL4159880 IC50 = 4242.0 nM 5.37
CHEMBL4174056 IC50 = 4400.0 nM 5.36
CHEMBL4169887 IC50 = 5361.0 nM 5.27
CHEMBL4162692 IC50 = 5775.0 nM 5.24
CHEMBL4166141 IC50 = 6010.0 nM 5.22
CHEMBL4172353 IC50 = 6090.0 nM 5.21
CHEMBL4174372 IC50 = 9115.0 nM 5.04
CHEMBL4160696 IC50 = 9070.0 nM 5.04
CHEMBL4101303 IC50 = 14295.0 nM 4.84
CHEMBL4101303 IC50 = 19925.0 nM 4.70
CHEMBL4163077 IC50 - -
CHEMBL4173902 IC50 > 10000.0 nM -
CHEMBL4165973 IC50 - -
CHEMBL4162121 IC50 > 10000.0 nM -
CHEMBL4159705 IC50 > 10000.0 nM -
CHEMBL4170331 IC50 > 10000.0 nM -
CHEMBL4169938 IC50 - -
CHEMBL4170940 IC50 > 10000.0 nM -
CHEMBL4170921 IC50 > 10000.0 nM -
CHEMBL4167954 IC50 > 10000.0 nM -
CHEMBL4175814 IC50 > 10000.0 nM -
CHEMBL4162281 IC50 > 10000.0 nM -
CHEMBL4172950 IC50 > 10000.0 nM -
CHEMBL4175003 IC50 - -
CHEMBL4174452 IC50 > 10000.0 nM -