Assay Detail
Binding
CHEMBL4149807
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of mu opioid receptor (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of N-Alkyl Piperazine Side Chain Based CXCR4 Antagonists with Improved Drug-like Properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.89 | 4.95 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4174290 | — | — | 1 | 4.95 |
| CHEMBL3091687 | — | — | 1 | 4.83 |
| CHEMBL4167058 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4174290 | — | IC50 | = | 11300.0 | nM | 4.95 |
| CHEMBL3091687 | — | IC50 | = | 14900.0 | nM | 4.83 |
| CHEMBL4167058 | — | IC50 | > | 30000.0 | nM | - |