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Assay Detail

CHEMBL4186904

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human DU145 cells after 48 hrs by MTT assay
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type DU-145
Confidence 1 — Organism
Curated By Intermediate

Target

DU-145 (CHEMBL613508)
Type CELL-LINE
Organism Homo sapiens

Publication

Podophyllotoxin derivatives as an excellent anticancer aspirant for future chemotherapy: A key current imminent needs.
Zhang X, Rakesh KP, Shantharam CS, Manukumar HM, Asiri AM, Marwani HM, Qin HL.
Bioorg Med Chem (2018) 26 : 340 -355
PubMed 29269253 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.87 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4214590 1 5.92
CHEMBL4205298 1 5.92
CHEMBL4216087 1 5.92
CHEMBL4217545 1 5.92
CHEMBL44657 ETOPOSIDE 4.0 1 5.69

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4214590 IC50 = 1200.0 nM 5.92
CHEMBL4205298 IC50 = 1200.0 nM 5.92
CHEMBL4216087 IC50 = 1200.0 nM 5.92
CHEMBL4217545 IC50 = 1200.0 nM 5.92
CHEMBL44657 ETOPOSIDE IC50 = 2030.0 nM 5.69