Assay Detail
Binding
CHEMBL4190750
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]DAMGO from mu opioid receptor in guinea pig brain membranes after 120 mins by scintillation counting analysis
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Tissue | Brain |
| Subcellular | Membrane |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 11 | 7.09 | 8.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL80 | NALOXONE | 4.0 | 1 | 8.68 |
| CHEMBL70 | MORPHINE | 4.0 | 1 | 8.41 |
| CHEMBL4206082 | — | — | 1 | 6.58 |
| CHEMBL4218965 | — | — | 1 | 6.35 |
| CHEMBL4216717 | — | — | 1 | 6.30 |
| CHEMBL4209225 | — | — | 1 | 6.20 |
| CHEMBL4216136 | — | — | 1 | - |
| CHEMBL4203850 | — | — | 1 | - |
| CHEMBL4203694 | — | — | 1 | - |
| CHEMBL4215892 | — | — | 1 | - |
| CHEMBL4212604 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL80 | NALOXONE | Ki | = | 2.1 | nM | 8.68 |
| CHEMBL70 | MORPHINE | Ki | = | 3.9 | nM | 8.41 |
| CHEMBL4206082 | — | Ki | = | 261.0 | nM | 6.58 |
| CHEMBL4218965 | — | Ki | = | 447.0 | nM | 6.35 |
| CHEMBL4216717 | — | Ki | = | 502.0 | nM | 6.30 |
| CHEMBL4209225 | — | Ki | = | 633.0 | nM | 6.20 |
| CHEMBL4216136 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL4203850 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL4203694 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL4215892 | — | Ki | > | 1000.0 | nM | - |
| CHEMBL4212604 | — | Ki | > | 1000.0 | nM | - |