Assay Detail
Binding
CHEMBL4197677
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Binding affinity to MOR (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Benzomorphan scaffold for opioid analgesics and pharmacological tools development: A comprehensive review.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.33 | 9.11 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL55033 | — | — | 1 | 9.11 |
| CHEMBL4218284 | — | — | 1 | 7.35 |
| CHEMBL4213351 | — | — | 1 | 5.54 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL55033 | — | Ki | = | 0.78 | nM | 9.11 |
| CHEMBL4218284 | — | Ki | = | 45.0 | nM | 7.35 |
| CHEMBL4213351 | — | Ki | = | 2900.0 | nM | 5.54 |