Assay Detail
Binding
CHEMBL4324467
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Displacement of 2-[125I]iodomelatonin from chick brain melatonin receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Gallus gallus |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Indole-based melatonin analogues: Synthetic approaches and biological activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.33 | 9.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL142343 | — | — | 1 | 9.42 |
| CHEMBL45 | MELATONIN | 4.0 | 1 | 9.23 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL142343 | — | Ki | = | 0.378 | nM | 9.42 |
| CHEMBL45 | MELATONIN | Ki | = | 0.59 | nM | 9.23 |