Assay Detail
Binding
CHEMBL4356409
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Competitive inhibition of UCHL1 in human H1299 cells using Ub-AMC substrate
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Ubiquitin carboxyl-terminal hydrolase isozyme L1 (CHEMBL6159) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Advances in Discovering Deubiquitinating Enzyme (DUB) Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.40 | 6.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3407553 | — | — | 1 | 6.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3407553 | — | Ki | = | 400.0 | nM | 6.40 |