Assay Detail
Functional
CHEMBL4356743
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human MOLM16 cells assessed as reduction in cell viability incubated for 4 days by cell-titer glo luminescent assay
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Structure-Based Discovery of SD-36 as a Potent, Selective, and Efficacious PROTAC Degrader of STAT3 Protein.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 25 | 6.70 | 7.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4452527 | — | — | 1 | 7.89 |
| CHEMBL4541088 | — | — | 1 | 7.60 |
| CHEMBL4469975 | — | — | 1 | 7.38 |
| CHEMBL4592058 | — | — | 1 | 7.23 |
| CHEMBL4546818 | — | — | 1 | 7.20 |
| CHEMBL4451225 | — | — | 1 | 7.17 |
| CHEMBL4552403 | — | — | 1 | 7.11 |
| CHEMBL4452301 | — | — | 1 | 7.04 |
| CHEMBL4589874 | — | — | 1 | 7.00 |
| CHEMBL4567496 | — | — | 1 | 6.98 |
| CHEMBL4462015 | — | — | 1 | 6.89 |
| CHEMBL4460570 | — | — | 1 | 6.83 |
| CHEMBL4561959 | — | — | 1 | 6.68 |
| CHEMBL4476035 | — | — | 1 | 6.65 |
| CHEMBL4593217 | — | — | 1 | 6.63 |
| CHEMBL4458633 | — | — | 1 | 6.62 |
| CHEMBL4455300 | — | — | 1 | 6.44 |
| CHEMBL4443577 | — | — | 1 | 6.24 |
| CHEMBL4585187 | — | — | 1 | 6.15 |
| CHEMBL4462902 | — | — | 1 | 6.02 |
| CHEMBL4513915 | — | — | 1 | 5.90 |
| CHEMBL4532980 | — | — | 1 | 5.28 |
| CHEMBL4575382 | — | — | 1 | 5.19 |
| CHEMBL4531706 | — | — | 1 | - |
| CHEMBL4465803 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4452527 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL4541088 | — | IC50 | = | 25.0 | nM | 7.60 |
| CHEMBL4469975 | — | IC50 | = | 42.0 | nM | 7.38 |
| CHEMBL4592058 | — | IC50 | = | 59.0 | nM | 7.23 |
| CHEMBL4546818 | — | IC50 | = | 63.0 | nM | 7.20 |
| CHEMBL4451225 | — | IC50 | = | 67.0 | nM | 7.17 |
| CHEMBL4552403 | — | IC50 | = | 78.0 | nM | 7.11 |
| CHEMBL4452301 | — | IC50 | = | 91.0 | nM | 7.04 |
| CHEMBL4589874 | — | IC50 | = | 99.0 | nM | 7.00 |
| CHEMBL4567496 | — | IC50 | = | 104.0 | nM | 6.98 |
| CHEMBL4462015 | — | IC50 | = | 128.0 | nM | 6.89 |
| CHEMBL4460570 | — | IC50 | = | 147.0 | nM | 6.83 |
| CHEMBL4561959 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL4476035 | — | IC50 | = | 226.0 | nM | 6.65 |
| CHEMBL4593217 | — | IC50 | = | 232.0 | nM | 6.63 |
| CHEMBL4458633 | — | IC50 | = | 241.0 | nM | 6.62 |
| CHEMBL4455300 | — | IC50 | = | 360.0 | nM | 6.44 |
| CHEMBL4443577 | — | IC50 | = | 582.0 | nM | 6.24 |
| CHEMBL4585187 | — | IC50 | = | 711.0 | nM | 6.15 |
| CHEMBL4462902 | — | IC50 | = | 950.0 | nM | 6.02 |
| CHEMBL4513915 | — | IC50 | = | 1250.0 | nM | 5.90 |
| CHEMBL4532980 | — | IC50 | = | 5210.0 | nM | 5.28 |
| CHEMBL4575382 | — | IC50 | = | 6450.0 | nM | 5.19 |
| CHEMBL4531706 | — | IC50 | > | 2000.0 | nM | - |
| CHEMBL4465803 | — | IC50 | > | 2000.0 | nM | - |