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Assay Detail

CHEMBL4384763

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Reversible inhibition of CYP3A4 (unknown origin) in presence of NADPH by vivid red substrate-based assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 3A4 (CHEMBL340)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Design and Optimization of Sulfone Pyrrolidine Sulfonamide Antagonists of Transient Receptor Potential Vanilloid-4 with in Vivo Activity in a Pulmonary Edema Model.
Pero JE, Matthews JM, Behm DJ, Brnardic EJ, Brooks C, Budzik BW, Costell MH, Donatelli CA, Eisennagel SH, Erhard K, Fischer MC, Holt DA, Jolivette LJ, Li H, Li P, McAtee JJ, McCleland BW, Pendrak I, Posobiec LM, Rivera KLK, Rivero RA, Roethke TJ, Sender MR, Shu A, Terrell LR, Vaidya K, Xu X, Lawhorn BG.
J Med Chem (2018) 61 : 11209 -11220
PubMed 30500190 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.31 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4456312 1 7.00
CHEMBL4547537 1 6.52
CHEMBL4461475 1 5.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4456312 IC50 = 100.0 nM 7.00
CHEMBL4547537 IC50 = 300.0 nM 6.52
CHEMBL4461475 IC50 = 4000.0 nM 5.40