Assay Detail
Functional
CHEMBL4418797
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human NCI-H1975 cells assessed as decrease in cell viability incubated for 72 hrs by CellTiter-Glo assay
35
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H1975 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Myc modulators and uses thereof
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 35 | 4.71 | 5.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4546151 | — | — | 1 | 5.57 |
| CHEMBL4462590 | — | — | 1 | 5.10 |
| CHEMBL4472238 | — | — | 1 | 4.90 |
| CHEMBL4573749 | — | — | 1 | 4.81 |
| CHEMBL4441910 | — | — | 1 | 4.76 |
| CHEMBL4571888 | — | — | 1 | 4.70 |
| CHEMBL4473046 | — | — | 1 | 4.55 |
| CHEMBL4435169 | — | — | 1 | 4.46 |
| CHEMBL4592867 | — | — | 1 | 4.34 |
| CHEMBL4460085 | — | — | 1 | 4.34 |
| CHEMBL4578105 | — | — | 1 | 4.25 |
| CHEMBL4437143 | — | — | 1 | - |
| CHEMBL4438510 | — | — | 1 | - |
| CHEMBL4448869 | — | — | 1 | - |
| CHEMBL4546028 | — | — | 1 | - |
| CHEMBL4436103 | — | — | 1 | - |
| CHEMBL4543327 | — | — | 1 | - |
| CHEMBL4463878 | — | — | 1 | - |
| CHEMBL4457623 | — | — | 1 | - |
| CHEMBL4574226 | — | — | 1 | - |
| CHEMBL4573018 | — | — | 1 | - |
| CHEMBL4463755 | — | — | 1 | - |
| CHEMBL4440351 | — | — | 1 | - |
| CHEMBL4464803 | — | — | 1 | - |
| CHEMBL4435325 | — | — | 1 | - |
| CHEMBL4569060 | — | — | 1 | - |
| CHEMBL4449302 | — | — | 1 | - |
| CHEMBL4439086 | — | — | 1 | - |
| CHEMBL4515991 | — | — | 1 | - |
| CHEMBL4456540 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4546151 | — | IC50 | = | 2713.0 | nM | 5.57 |
| CHEMBL4462590 | — | IC50 | = | 7880.0 | nM | 5.10 |
| CHEMBL4472238 | — | IC50 | = | 12470.0 | nM | 4.90 |
| CHEMBL4573749 | — | IC50 | = | 15580.0 | nM | 4.81 |
| CHEMBL4441910 | — | IC50 | = | 17320.0 | nM | 4.76 |
| CHEMBL4571888 | — | IC50 | = | 19950.0 | nM | 4.70 |
| CHEMBL4473046 | — | IC50 | = | 28180.0 | nM | 4.55 |
| CHEMBL4435169 | — | IC50 | = | 34530.0 | nM | 4.46 |
| CHEMBL4592867 | — | IC50 | = | 45270.0 | nM | 4.34 |
| CHEMBL4460085 | — | IC50 | = | 45310.0 | nM | 4.34 |
| CHEMBL4578105 | — | IC50 | = | 56300.0 | nM | 4.25 |
| CHEMBL4463878 | — | IC50 | - | — | - | |
| CHEMBL4543327 | — | IC50 | - | — | - | |
| CHEMBL4436103 | — | IC50 | - | — | - | |
| CHEMBL4546028 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4448869 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4438510 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4437143 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4564939 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4459178 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4591315 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4448611 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4574522 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL4457623 | — | IC50 | - | — | - | |
| CHEMBL4574226 | — | IC50 | - | — | - | |
| CHEMBL4573018 | — | IC50 | - | — | - | |
| CHEMBL4463755 | — | IC50 | - | — | - | |
| CHEMBL4440351 | — | IC50 | - | — | - | |
| CHEMBL4464803 | — | IC50 | - | — | - | |
| CHEMBL4435325 | — | IC50 | - | — | - | |
| CHEMBL4569060 | — | IC50 | - | — | - | |
| CHEMBL4449302 | — | IC50 | - | — | - | |
| CHEMBL4439086 | — | IC50 | - | — | - | |
| CHEMBL4515991 | — | IC50 | - | — | - | |
| CHEMBL4456540 | — | IC50 | - | — | - |