Assay Detail
Binding
CHEMBL4419259
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to AKT PH-domain (unknown origin) at 0.01 to 50 uM by SPR spectroscopy
37
Total Activities
37
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
RAC-alpha serine/threonine-protein kinase (CHEMBL4282) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Methods and compositions for inhibiting cnksr1
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 30 | 5.25 | 9.32 |
| Activity | 7 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL244695 | — | — | 1 | 9.32 |
| CHEMBL4576938 | — | — | 1 | 5.60 |
| CHEMBL4464276 | — | — | 1 | 5.60 |
| CHEMBL4439996 | — | — | 1 | 5.32 |
| CHEMBL4437164 | — | — | 1 | 5.21 |
| CHEMBL4451129 | — | — | 1 | 4.87 |
| CHEMBL1422005 | — | — | 1 | 4.76 |
| CHEMBL4542842 | — | — | 1 | 4.47 |
| CHEMBL4446354 | — | — | 1 | 4.29 |
| CHEMBL4528582 | — | — | 1 | 4.18 |
| CHEMBL4293794 | — | — | 1 | 4.12 |
| CHEMBL4441334 | — | — | 1 | - |
| CHEMBL4540854 | — | — | 1 | - |
| CHEMBL4557494 | — | — | 1 | - |
| CHEMBL4526378 | — | — | 1 | - |
| CHEMBL4527518 | — | — | 1 | - |
| CHEMBL2030270 | — | — | 1 | - |
| CHEMBL4472901 | — | — | 1 | - |
| CHEMBL4280751 | — | — | 1 | - |
| CHEMBL4280394 | — | — | 1 | - |
| CHEMBL4552253 | — | — | 1 | - |
| CHEMBL4279325 | — | — | 1 | - |
| CHEMBL4442523 | — | — | 1 | - |
| CHEMBL4283567 | — | — | 1 | - |
| CHEMBL4287230 | — | — | 1 | - |
| CHEMBL4451466 | — | — | 1 | - |
| CHEMBL4588492 | — | — | 1 | - |
| CHEMBL4529653 | — | — | 1 | - |
| CHEMBL4515226 | — | — | 1 | - |
| CHEMBL4473695 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL244695 | — | Kd | = | 0.474 | nM | 9.32 |
| CHEMBL4576938 | — | Kd | = | 2530.0 | nM | 5.60 |
| CHEMBL4464276 | — | Kd | = | 2530.0 | nM | 5.60 |
| CHEMBL4439996 | — | Kd | = | 4800.0 | nM | 5.32 |
| CHEMBL4437164 | — | Kd | = | 6220.0 | nM | 5.21 |
| CHEMBL4451129 | — | Kd | = | 13500.0 | nM | 4.87 |
| CHEMBL1422005 | — | Kd | = | 17300.0 | nM | 4.76 |
| CHEMBL4542842 | — | Kd | = | 34200.0 | nM | 4.47 |
| CHEMBL4446354 | — | Kd | = | 51600.0 | nM | 4.29 |
| CHEMBL4528582 | — | Kd | = | 66300.0 | nM | 4.18 |
| CHEMBL4293794 | — | Kd | = | 75200.0 | nM | 4.12 |
| CHEMBL2030270 | — | Activity | - | — | - | |
| CHEMBL4542845 | — | Kd | - | — | - | |
| CHEMBL4527518 | — | Activity | - | — | - | |
| CHEMBL4526378 | — | Activity | - | — | - | |
| CHEMBL4557494 | — | Activity | - | — | - | |
| CHEMBL4540854 | — | Activity | - | — | - | |
| CHEMBL4441334 | — | Activity | - | — | - | |
| CHEMBL4579008 | — | Kd | = | 0.00128 | nM | - |
| CHEMBL4482955 | — | Kd | - | — | - | |
| CHEMBL4519349 | — | Kd | - | — | - | |
| CHEMBL4435105 | — | Kd | - | — | - | |
| CHEMBL4465082 | — | Kd | - | — | - | |
| CHEMBL4533907 | — | Kd | - | — | - | |
| CHEMBL4472901 | — | Kd | - | — | - | |
| CHEMBL4280751 | — | Kd | - | — | - | |
| CHEMBL4280394 | — | Kd | > | 500000.0 | nM | - |
| CHEMBL4552253 | — | Kd | = | 178000.0 | nM | - |
| CHEMBL4279325 | — | Kd | > | 500000.0 | nM | - |
| CHEMBL4442523 | — | Kd | - | — | - | |
| CHEMBL4283567 | — | Kd | - | — | - | |
| CHEMBL4287230 | — | Kd | - | — | - | |
| CHEMBL4451466 | — | Kd | = | 330000.0 | nM | - |
| CHEMBL4588492 | — | Activity | - | — | - | |
| CHEMBL4529653 | — | Kd | = | 286000.0 | nM | - |
| CHEMBL4515226 | — | Kd | = | 133000.0 | nM | - |
| CHEMBL4473695 | — | Kd | = | 140000.0 | nM | - |