Assay Detail
Binding
CHEMBL4422548
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of GST-fused human Eya2 ED (253 to 538 residues) expressed in Escherichia coli pre-incubated for 10 mins before phosphorylated H2AX peptide substrate addition and further incubated for 40 mins by malachite green-based secondary phosphatase assay
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Inhibitors of eya2
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 4.76 | 4.78 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4459891 | — | — | 1 | 4.78 |
| CHEMBL1975051 | — | — | 1 | 4.78 |
| CHEMBL3195222 | — | — | 1 | 4.78 |
| CHEMBL4445513 | — | — | 1 | 4.78 |
| CHEMBL3189517 | — | — | 1 | 4.78 |
| CHEMBL3190554 | — | — | 1 | 4.78 |
| CHEMBL4446792 | — | — | 1 | 4.78 |
| CHEMBL4476815 | — | — | 1 | 4.78 |
| CHEMBL4446652 | — | — | 1 | 4.78 |
| CHEMBL3191598 | — | — | 1 | 4.78 |
| CHEMBL4530754 | — | — | 1 | 4.78 |
| CHEMBL4458563 | — | — | 1 | 4.74 |
| CHEMBL4532983 | — | — | 1 | 4.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4459891 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL1975051 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL3195222 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL4445513 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL3189517 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL3190554 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL4446792 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL4476815 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL4446652 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL3191598 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL4530754 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL4458563 | — | IC50 | = | 18250.0 | nM | 4.74 |
| CHEMBL4532983 | — | IC50 | = | 31980.0 | nM | 4.50 |