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Assay Detail

CHEMBL4425908

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of CYP3A4 (unknown origin)
11
Total Activities
11
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 3A4 (CHEMBL340)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Discovery of (S)-1-(1-(4-Chloro-3-fluorophenyl)-2-hydroxyethyl)-4-(2-((1-methyl-1H-pyrazol-5-yl)amino)pyrimidin-4-yl)pyridin-2(1H)-one (GDC-0994), an Extracellular Signal-Regulated Kinase 1/2 (ERK1/2) Inhibitor in Early Clinical Development.
Blake JF, Burkard M, Chan J, Chen H, Chou KJ, Diaz D, Dudley DA, Gaudino JJ, Gould SE, Grina J, Hunsaker T, Liu L, Martinson M, Moreno D, Mueller L, Orr C, Pacheco P, Qin A, Rasor K, Ren L, Robarge K, Shahidi-Latham S, Stults J, Sullivan F, Wang W, Yin J, Zhou A, Belvin M, Merchant M, Moffat J, Schwarz JB.
J Med Chem (2016) 59 : 5650 -5660
PubMed 27227380 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Inhibition 10 - -
IC50 1 6.47 6.47

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4571067 1 6.47
CHEMBL4435650 1 -
CHEMBL4592894 1 -
CHEMBL4114404 1 -
CHEMBL4460988 1 -
CHEMBL3675721 1 -
CHEMBL4436718 1 -
CHEMBL4474917 1 -
CHEMBL4565958 1 -
CHEMBL4527526 1 -
CHEMBL4446409 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4571067 IC50 = 340.0 nM 6.47
CHEMBL4435650 Inhibition - % -
CHEMBL4592894 Inhibition - % -
CHEMBL4114404 Inhibition - % -
CHEMBL4460988 Inhibition - % -
CHEMBL3675721 Inhibition - % -
CHEMBL4436718 Inhibition - % -
CHEMBL4474917 Inhibition - % -
CHEMBL4565958 Inhibition - % -
CHEMBL4527526 Inhibition - % -
CHEMBL4446409 Inhibition - % -