Assay Detail
Functional
CHEMBL4613567
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Antiproliferative activity against human HL60 cells after 72 hrs by MTT assay
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Quinolone hybrids and their anti-cancer activities: An overview.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 7.52 | 7.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4645895 | — | — | 1 | 7.75 |
| CHEMBL4633435 | — | — | 1 | 7.50 |
| CHEMBL4647394 | — | — | 1 | 7.50 |
| CHEMBL4636122 | — | — | 1 | 7.50 |
| CHEMBL4649384 | — | — | 1 | 7.50 |
| CHEMBL4647558 | — | — | 1 | 7.50 |
| CHEMBL4640038 | — | — | 1 | 7.50 |
| CHEMBL4640200 | — | — | 1 | 7.50 |
| CHEMBL4632631 | — | — | 1 | 7.50 |
| CHEMBL4638094 | — | — | 1 | 7.50 |
| CHEMBL4637492 | — | — | 1 | 7.50 |
| CHEMBL4634909 | — | — | 1 | 7.50 |
| CHEMBL4636149 | — | — | 1 | 7.50 |
| CHEMBL4633427 | — | — | 1 | 7.50 |
| CHEMBL4639575 | — | — | 1 | 7.50 |
| CHEMBL481 | IRINOTECAN | 4.0 | 1 | 7.50 |
| CHEMBL8 | CIPROFLOXACIN | 4.0 | 1 | - |
| CHEMBL9 | NORFLOXACIN | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4645895 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL4633435 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4647394 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4636122 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4649384 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4647558 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4640038 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4640200 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4632631 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4638094 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4637492 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4634909 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4636149 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4633427 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4639575 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL481 | IRINOTECAN | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL8 | CIPROFLOXACIN | IC50 | > | 302.0 | nM | - |
| CHEMBL9 | NORFLOXACIN | IC50 | > | 302.0 | nM | - |