Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL4616761

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against mouse B16F10 cells assessed as reduction in cell viability
39
Total Activities
39
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type B16-F10
Confidence 1 — Organism
Curated By Autocuration

Target

B16-F10 (CHEMBL612656)
Type CELL-LINE
Organism Mus musculus

Publication

Green recipes to quinoline: A review.
Nainwal LM, Tasneem S, Akhtar W, Verma G, Khan MF, Parvez S, Shaquiquzzaman M, Akhter M, Alam MM.
Eur J Med Chem (2019) 164 : 121 -170
PubMed 30594028 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 39 4.15 4.15

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1442731 1 4.15
CHEMBL4641258 1 4.15
CHEMBL4639632 1 4.15
CHEMBL4635111 1 4.15
CHEMBL4643287 1 4.15
CHEMBL4639590 1 4.15
CHEMBL4642273 1 4.15
CHEMBL4649856 1 4.15
CHEMBL2032372 1 4.15
CHEMBL4648126 1 4.15
CHEMBL4641143 1 4.15
CHEMBL3985661 1 4.15
CHEMBL3265260 1 4.15
CHEMBL2228156 2-CHLORONICOTINALDEHYDE 1 4.15
CHEMBL274794 2-PYRIDINECARBOXALDEHYDE 1 4.15
CHEMBL3753357 1 4.15
CHEMBL1531235 1 4.15
CHEMBL4645306 1 4.15
CHEMBL3236916 1 4.15
CHEMBL1568619 1 4.15
CHEMBL4646712 1 4.15
CHEMBL1474 1 4.15
CHEMBL3183207 1 4.15
CHEMBL4473405 1 4.15
CHEMBL164236 1 4.15
CHEMBL190927 1 4.15
CHEMBL14193 4-HYDROXYBENZALDEHYDE 1 4.15
CHEMBL161598 ANISALDEHYDE 1 4.15
CHEMBL15972 BENZALDEHYDE -1.0 1 4.15
CHEMBL4636372 1 4.15

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4641258 IC50 = 70740.0 nM 4.15
CHEMBL4641143 IC50 = 70740.0 nM 4.15
CHEMBL4648126 IC50 = 70740.0 nM 4.15
CHEMBL2032372 IC50 = 70740.0 nM 4.15
CHEMBL4649856 IC50 = 70740.0 nM 4.15
CHEMBL4642273 IC50 = 70740.0 nM 4.15
CHEMBL4639590 IC50 = 70740.0 nM 4.15
CHEMBL4643287 IC50 = 70740.0 nM 4.15
CHEMBL4635111 IC50 = 70740.0 nM 4.15
CHEMBL4639632 IC50 = 70740.0 nM 4.15
CHEMBL3985661 IC50 = 70740.0 nM 4.15
CHEMBL301141 4-HYDROXYCOUMARINS IC50 = 70740.0 nM 4.15
CHEMBL4647406 IC50 = 70740.0 nM 4.15
CHEMBL4638140 IC50 = 70740.0 nM 4.15
CHEMBL4648744 IC50 = 70740.0 nM 4.15
CHEMBL4639159 IC50 = 70740.0 nM 4.15
CHEMBL4649353 IC50 = 70740.0 nM 4.15
CHEMBL4638061 IC50 = 70740.0 nM 4.15
CHEMBL4632388 IC50 = 70740.0 nM 4.15
CHEMBL4642303 IC50 = 70740.0 nM 4.15
CHEMBL4646712 IC50 = 70740.0 nM 4.15
CHEMBL4636372 IC50 = 70740.0 nM 4.15
CHEMBL15972 BENZALDEHYDE IC50 = 70740.0 nM 4.15
CHEMBL161598 ANISALDEHYDE IC50 = 70740.0 nM 4.15
CHEMBL14193 4-HYDROXYBENZALDEHYDE IC50 = 70740.0 nM 4.15
CHEMBL190927 IC50 = 70740.0 nM 4.15
CHEMBL164236 IC50 = 70740.0 nM 4.15
CHEMBL4473405 IC50 = 70740.0 nM 4.15
CHEMBL3183207 IC50 = 70740.0 nM 4.15
CHEMBL1474 IC50 = 70740.0 nM 4.15
CHEMBL3753357 IC50 = 70740.0 nM 4.15
CHEMBL1568619 IC50 = 70740.0 nM 4.15
CHEMBL3236916 IC50 = 70740.0 nM 4.15
CHEMBL4645306 IC50 = 70740.0 nM 4.15
CHEMBL1531235 IC50 = 70740.0 nM 4.15
CHEMBL1442731 IC50 = 70740.0 nM 4.15
CHEMBL274794 2-PYRIDINECARBOXALDEHYDE IC50 = 70740.0 nM 4.15
CHEMBL2228156 2-CHLORONICOTINALDEHYDE IC50 = 70740.0 nM 4.15
CHEMBL3265260 IC50 = 70740.0 nM 4.15