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Assay Detail

CHEMBL4622623

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Ebolavirus infected in human HeLa cells assessed as reduction in viral replication incubated for 48 hrs by luminescence based assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Ebolavirus
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

Ebolavirus (CHEMBL4434621)
Type ORGANISM
Organism Ebolavirus

Publication

Toward the Target: Tilorone, Quinacrine, and Pyronaridine Bind to Ebola Virus Glycoprotein.
Lane TR, Ekins S.
ACS Med Chem Lett (2020) 11 : 1653 -1658
PubMed 32832035 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.00 6.09

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL35228 PYRONARIDINE 3.0 1 6.09
CHEMBL7568 QUINACRINE 4.0 1 5.98
CHEMBL47298 TILORONE 2.0 1 5.94

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL35228 PYRONARIDINE IC50 = 820.0 nM 6.09
CHEMBL7568 QUINACRINE IC50 = 1050.0 nM 5.98
CHEMBL47298 TILORONE IC50 = 1140.0 nM 5.94