Assay Detail
Functional
CHEMBL4825887
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Antiviral activity against Respiratory syncytial virus A2 infected in African green monkey Vero cells by Plaque reduction assay
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Human respiratory syncytial virus |
| Cell Type | Vero |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of Sisunatovir (RV521), an Inhibitor of Respiratory Syncytial Virus Fusion.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 21 | 6.86 | 9.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4878302 | — | — | 1 | 9.10 |
| CHEMBL4297497 | SISUNATOVIR | 2.0 | 1 | 8.89 |
| CHEMBL4872095 | — | — | 1 | 8.38 |
| CHEMBL4876843 | — | — | 1 | 8.27 |
| CHEMBL4865906 | — | — | 1 | 8.17 |
| CHEMBL4859694 | — | — | 1 | 7.75 |
| CHEMBL4872263 | — | — | 1 | 7.59 |
| CHEMBL4469438 | — | — | 1 | 7.51 |
| CHEMBL4860271 | — | — | 1 | 7.39 |
| CHEMBL4862291 | — | — | 1 | 6.74 |
| CHEMBL4845727 | — | — | 1 | 6.62 |
| CHEMBL4877602 | — | — | 1 | 6.51 |
| CHEMBL4850153 | — | — | 1 | 6.35 |
| CHEMBL4869353 | — | — | 1 | 6.34 |
| CHEMBL4874044 | — | — | 1 | 6.24 |
| CHEMBL4855486 | — | — | 1 | 5.77 |
| CHEMBL4878086 | — | — | 1 | 5.62 |
| CHEMBL4851012 | — | — | 1 | 5.47 |
| CHEMBL4873987 | — | — | 1 | 5.44 |
| CHEMBL4878851 | — | — | 1 | 4.99 |
| CHEMBL4868500 | — | — | 1 | 4.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4878302 | — | EC50 | = | 0.8 | nM | 9.10 |
| CHEMBL4297497 | SISUNATOVIR | EC50 | = | 1.3 | nM | 8.89 |
| CHEMBL4872095 | — | EC50 | = | 4.2 | nM | 8.38 |
| CHEMBL4876843 | — | EC50 | = | 5.4 | nM | 8.27 |
| CHEMBL4865906 | — | EC50 | = | 6.7 | nM | 8.17 |
| CHEMBL4859694 | — | EC50 | = | 17.9 | nM | 7.75 |
| CHEMBL4872263 | — | EC50 | = | 25.4 | nM | 7.59 |
| CHEMBL4469438 | — | EC50 | = | 31.0 | nM | 7.51 |
| CHEMBL4860271 | — | EC50 | = | 40.8 | nM | 7.39 |
| CHEMBL4862291 | — | EC50 | = | 180.7 | nM | 6.74 |
| CHEMBL4845727 | — | EC50 | = | 240.0 | nM | 6.62 |
| CHEMBL4877602 | — | EC50 | = | 310.0 | nM | 6.51 |
| CHEMBL4850153 | — | EC50 | = | 444.2 | nM | 6.35 |
| CHEMBL4869353 | — | EC50 | = | 453.9 | nM | 6.34 |
| CHEMBL4874044 | — | EC50 | = | 580.0 | nM | 6.24 |
| CHEMBL4855486 | — | EC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL4878086 | — | EC50 | = | 2384.3 | nM | 5.62 |
| CHEMBL4851012 | — | EC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL4873987 | — | EC50 | = | 3636.0 | nM | 5.44 |
| CHEMBL4878851 | — | EC50 | = | 10181.3 | nM | 4.99 |
| CHEMBL4868500 | — | EC50 | = | 14000.0 | nM | 4.85 |