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Compound Detail

CHEMBL4874044

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CC(C)CCn1c(CN2C(=O)C3(CCCC3)c3ccccc32)nc2cc(CN)ccc21

Basic Information

ChEMBL ID CHEMBL4874044
Phase Preclinical
Structure Type MOL
InChI Key OHLCUWXCUOAYGO-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

416.6
MW (Da)
4.90
ALogP
4
HBA
1
HBD
64.2
PSA (Ų)
0.62
QED
0
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C26H32N4O
MW 416.57
Aromatic Rings 3
Heavy Atoms 31
NP-Likeness -0.89

Activity Summary

EC50 1 meas. best 6.24

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human orthopneumovirus
CHEMBL613127
EC50 6.24 6.24 580.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
33729773 10.1021/acs.jmedchem.0c01882 Human orthopneumovirus 1
33729773 10.1021/acs.jmedchem.0c01882 Vero 1

Data from ChEMBL 36 via Core Engine