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Assay Detail

CHEMBL4840652

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Trypanocidal activity against Trypanosoma cruzi amastigotes assessed as inhibition of parasite growth by alamar blue staining based fluorescence analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Trypanosoma cruzi
Confidence 1 — Organism
Curated By Autocuration

Target

Trypanosoma cruzi (CHEMBL368)
Type ORGANISM
Organism Trypanosoma cruzi

Publication

Design and synthesis of Mannich base-type derivatives containing imidazole and benzimidazole as lead compounds for drug discovery in Chagas Disease.
Beltran-Hortelano I, Atherton RL, Rubio-Hernández M, Sanz-Serrano J, Alcolea V, Kelly JM, Pérez-Silanes S, Olmo F.
Eur J Med Chem (2021) 223 : 113646 -113646
PubMed 34182359 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.40 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4856014 1 6.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4856014 IC50 = 400.0 nM 6.40