Assay Detail
Functional
CHEMBL4883190
Review assay metadata, readout intent, target linkage, and publication context from the same page.
CHO-based cAMP assay (human)
2
Total Activities
2
Compounds Tested
1
Activity Types
2
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe TP-024
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 7.03 | 7.03 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Assay publication | Assay publication | - | — | PMID: 28433511 |
| Target protein type | Target protein type | - | — | GPR52 expressed CHO cell line |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4082756 | TP-024 | — | 1 | 7.03 |
| CHEMBL4100408 | TP-024n | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4082756 | TP-024 | EC50 | = | 93.0 | nM | 7.03 |
| CHEMBL4100408 | TP-024n | EC50 | > | 1000.0 | nM | - |