Assay Detail
Binding
CHEMBL5127643
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Inhibition of MOP (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Analgesic Opioid Ligand Discovery Based on Nonmorphinan Scaffolds Derived from Natural Sources.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.43 | 5.66 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4848517 | — | — | 1 | 5.66 |
| CHEMBL4546925 | — | — | 1 | 5.38 |
| CHEMBL4859858 | — | — | 1 | 5.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4848517 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL4546925 | — | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL4859858 | — | IC50 | = | 5700.0 | nM | 5.24 |