Assay Detail
Binding
CHEMBL5140913
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Binding affinity to rat Androgen receptor
3
Total Activities
3
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Therapeutic Strategies to Target the Androgen Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.74 | 7.89 |
| Ki | 1 | 8.21 | 8.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL197595 | — | — | 1 | 8.21 |
| CHEMBL1684194 | — | — | 1 | 7.89 |
| CHEMBL1910411 | — | — | 1 | 7.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL197595 | — | Ki | = | 6.2 | nM | 8.21 |
| CHEMBL1684194 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL1910411 | — | IC50 | = | 26.0 | nM | 7.58 |