Assay Detail
Functional
CHEMBL5217430
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Anticancer activity against human SK-N-AS cells assessed as reduction in cell viability incubated for 48 hrs by resazurin dye based fluorescence assay
15
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | SK-N-AS |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Multiple approaches to repurposing drugs for neuroblastoma.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.40 | 5.91 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL403183 | — | — | 1 | 5.91 |
| CHEMBL1448 | NICLOSAMIDE | 4.0 | 1 | 5.63 |
| CHEMBL35228 | PYRONARIDINE | 3.0 | 1 | 5.46 |
| CHEMBL1818132 | — | — | 1 | 5.41 |
| CHEMBL1983268 | ENTRECTINIB | 4.0 | 1 | 5.35 |
| CHEMBL5220528 | — | — | 1 | 5.27 |
| CHEMBL314854 | FINGOLIMOD | 4.0 | 1 | 5.21 |
| CHEMBL601719 | CRIZOTINIB | 4.0 | 1 | 4.92 |
| CHEMBL5219915 | — | — | 1 | - |
| CHEMBL5219687 | — | — | 1 | - |
| CHEMBL5218687 | — | — | 1 | - |
| CHEMBL588079 | — | — | 1 | - |
| CHEMBL5219722 | — | — | 1 | - |
| CHEMBL5221024 | — | — | 1 | - |
| CHEMBL7568 | QUINACRINE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL403183 | — | IC50 | = | 1230.0 | nM | 5.91 |
| CHEMBL1448 | NICLOSAMIDE | IC50 | = | 2330.0 | nM | 5.63 |
| CHEMBL35228 | PYRONARIDINE | IC50 | = | 3450.0 | nM | 5.46 |
| CHEMBL1818132 | — | IC50 | = | 3860.0 | nM | 5.41 |
| CHEMBL1983268 | ENTRECTINIB | IC50 | = | 4470.0 | nM | 5.35 |
| CHEMBL5220528 | — | IC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL314854 | FINGOLIMOD | IC50 | = | 6110.0 | nM | 5.21 |
| CHEMBL601719 | CRIZOTINIB | IC50 | = | 12120.0 | nM | 4.92 |
| CHEMBL5219915 | — | IC50 | - | — | - | |
| CHEMBL5219687 | — | IC50 | - | — | - | |
| CHEMBL5218687 | — | IC50 | - | — | - | |
| CHEMBL588079 | — | IC50 | - | — | - | |
| CHEMBL5219722 | — | IC50 | - | — | - | |
| CHEMBL5221024 | — | IC50 | - | — | - | |
| CHEMBL7568 | QUINACRINE | IC50 | - | — | - |