Assay Detail
Functional
CHEMBL5226216
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human KARPAS-422 cell assessed as cell growth inhibition incubated for 6 days by ATPlite reagent based luminescence assay
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | KARPAS-422 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of OICR12694: A Novel, Potent, Selective, and Orally Bioavailable BCL6 BTB Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 34 | 6.57 | 8.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5282647 | — | — | 1 | 8.05 |
| CHEMBL5283745 | — | — | 1 | 7.89 |
| CHEMBL5270031 | — | — | 1 | 7.58 |
| CHEMBL5285804 | — | — | 1 | 7.19 |
| CHEMBL5275407 | — | — | 1 | 7.07 |
| CHEMBL5279363 | — | — | 1 | 7.04 |
| CHEMBL5269780 | — | — | 1 | 6.99 |
| CHEMBL5287446 | — | — | 1 | 6.92 |
| CHEMBL5288796 | — | — | 1 | 6.86 |
| CHEMBL5285971 | — | — | 1 | 6.85 |
| CHEMBL5269124 | — | — | 1 | 6.82 |
| CHEMBL5279982 | — | — | 1 | 6.79 |
| CHEMBL5291358 | — | — | 1 | 6.78 |
| CHEMBL5288047 | — | — | 1 | 6.70 |
| CHEMBL5271863 | — | — | 1 | 6.70 |
| CHEMBL5271784 | — | — | 1 | 6.68 |
| CHEMBL5287071 | — | — | 1 | 6.64 |
| CHEMBL5271042 | — | — | 1 | 6.57 |
| CHEMBL5268066 | — | — | 1 | 6.52 |
| CHEMBL5291478 | — | — | 1 | 6.39 |
| CHEMBL5290428 | — | — | 1 | 6.36 |
| CHEMBL5272054 | — | — | 1 | 6.34 |
| CHEMBL5276120 | — | — | 1 | 6.21 |
| CHEMBL5271895 | — | — | 1 | 6.19 |
| CHEMBL5285053 | — | — | 1 | 6.11 |
| CHEMBL5267067 | — | — | 1 | 6.10 |
| CHEMBL5279858 | — | — | 1 | 6.01 |
| CHEMBL5279299 | — | — | 1 | 5.96 |
| CHEMBL5284699 | — | — | 1 | 5.96 |
| CHEMBL5267621 | — | — | 1 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5282647 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL5283745 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL5270031 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL5285804 | — | IC50 | = | 65.0 | nM | 7.19 |
| CHEMBL5275407 | — | IC50 | = | 86.0 | nM | 7.07 |
| CHEMBL5279363 | — | IC50 | = | 92.0 | nM | 7.04 |
| CHEMBL5269780 | — | IC50 | = | 102.0 | nM | 6.99 |
| CHEMBL5287446 | — | IC50 | = | 119.0 | nM | 6.92 |
| CHEMBL5288796 | — | IC50 | = | 139.0 | nM | 6.86 |
| CHEMBL5285971 | — | IC50 | = | 142.0 | nM | 6.85 |
| CHEMBL5269124 | — | IC50 | = | 152.0 | nM | 6.82 |
| CHEMBL5279982 | — | IC50 | = | 162.0 | nM | 6.79 |
| CHEMBL5291358 | — | IC50 | = | 166.0 | nM | 6.78 |
| CHEMBL5288047 | — | IC50 | = | 202.0 | nM | 6.70 |
| CHEMBL5271863 | — | IC50 | = | 202.0 | nM | 6.70 |
| CHEMBL5271784 | — | IC50 | = | 207.0 | nM | 6.68 |
| CHEMBL5287071 | — | IC50 | = | 231.0 | nM | 6.64 |
| CHEMBL5271042 | — | IC50 | = | 270.0 | nM | 6.57 |
| CHEMBL5268066 | — | IC50 | = | 299.0 | nM | 6.52 |
| CHEMBL5291478 | — | IC50 | = | 407.0 | nM | 6.39 |
| CHEMBL5290428 | — | IC50 | = | 439.0 | nM | 6.36 |
| CHEMBL5272054 | — | IC50 | = | 457.0 | nM | 6.34 |
| CHEMBL5276120 | — | IC50 | = | 612.0 | nM | 6.21 |
| CHEMBL5271895 | — | IC50 | = | 644.0 | nM | 6.19 |
| CHEMBL5285053 | — | IC50 | = | 781.0 | nM | 6.11 |
| CHEMBL5267067 | — | IC50 | = | 796.0 | nM | 6.10 |
| CHEMBL5279858 | — | IC50 | = | 971.0 | nM | 6.01 |
| CHEMBL5279299 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL5284699 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL5267621 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL5286712 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL5286263 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL5284819 | — | IC50 | = | 7800.0 | nM | 5.11 |
| CHEMBL5267171 | — | IC50 | > | 10000.0 | nM | - |