Assay Detail
Binding
CHEMBL5318947
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of JNK1 (unknown origin) using ULight-4E-BP1 peptide as substrate incubated for 90 mins in presence of ATP by Lance ultra assay
68
Total Activities
68
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of Novel Indazole Chemotypes as Isoform-Selective JNK3 Inhibitors for the Treatment of Parkinson's Disease.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 68 | 5.13 | 7.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL252761 | — | — | 1 | 7.37 |
| CHEMBL5411091 | — | — | 1 | 5.14 |
| CHEMBL5437584 | — | — | 1 | 5.13 |
| CHEMBL5428091 | — | — | 1 | 5.12 |
| CHEMBL5402580 | — | — | 1 | 5.12 |
| CHEMBL5411375 | — | — | 1 | 5.12 |
| CHEMBL5403784 | — | — | 1 | 5.12 |
| CHEMBL5405579 | — | — | 1 | 5.12 |
| CHEMBL5439708 | — | — | 1 | 5.11 |
| CHEMBL5435391 | — | — | 1 | 5.11 |
| CHEMBL5403866 | — | — | 1 | 5.11 |
| CHEMBL5408361 | — | — | 1 | 5.11 |
| CHEMBL5408918 | — | — | 1 | 5.11 |
| CHEMBL5437979 | — | — | 1 | 5.11 |
| CHEMBL5423687 | — | — | 1 | 5.11 |
| CHEMBL5437251 | — | — | 1 | 5.11 |
| CHEMBL5432287 | — | — | 1 | 5.11 |
| CHEMBL5436065 | — | — | 1 | 5.10 |
| CHEMBL5409834 | — | — | 1 | 5.10 |
| CHEMBL5439622 | — | — | 1 | 5.09 |
| CHEMBL5433156 | — | — | 1 | 5.09 |
| CHEMBL5433711 | — | — | 1 | 5.08 |
| CHEMBL5441124 | — | — | 1 | 5.08 |
| CHEMBL5437898 | — | — | 1 | 5.07 |
| CHEMBL5398897 | — | — | 1 | 5.07 |
| CHEMBL5397012 | — | — | 1 | 5.07 |
| CHEMBL5428502 | — | — | 1 | 5.07 |
| CHEMBL5434414 | — | — | 1 | 5.07 |
| CHEMBL5413820 | — | — | 1 | 5.06 |
| CHEMBL5434519 | — | — | 1 | 5.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL252761 | — | IC50 | = | 42.34 | nM | 7.37 |
| CHEMBL5411091 | — | IC50 | = | 7247.0 | nM | 5.14 |
| CHEMBL5437584 | — | IC50 | = | 7412.0 | nM | 5.13 |
| CHEMBL5428091 | — | IC50 | = | 7682.0 | nM | 5.12 |
| CHEMBL5402580 | — | IC50 | = | 7593.0 | nM | 5.12 |
| CHEMBL5411375 | — | IC50 | = | 7673.0 | nM | 5.12 |
| CHEMBL5403784 | — | IC50 | = | 7659.0 | nM | 5.12 |
| CHEMBL5405579 | — | IC50 | = | 7612.0 | nM | 5.12 |
| CHEMBL5403866 | — | IC50 | = | 7819.0 | nM | 5.11 |
| CHEMBL5435391 | — | IC50 | = | 7698.0 | nM | 5.11 |
| CHEMBL5439708 | — | IC50 | = | 7791.0 | nM | 5.11 |
| CHEMBL5408361 | — | IC50 | = | 7745.0 | nM | 5.11 |
| CHEMBL5432287 | — | IC50 | = | 7703.0 | nM | 5.11 |
| CHEMBL5408918 | — | IC50 | = | 7703.0 | nM | 5.11 |
| CHEMBL5437979 | — | IC50 | = | 7686.0 | nM | 5.11 |
| CHEMBL5423687 | — | IC50 | = | 7803.0 | nM | 5.11 |
| CHEMBL5437251 | — | IC50 | = | 7843.0 | nM | 5.11 |
| CHEMBL5436065 | — | IC50 | = | 8018.0 | nM | 5.10 |
| CHEMBL5409834 | — | IC50 | = | 7998.0 | nM | 5.10 |
| CHEMBL5439622 | — | IC50 | = | 8207.0 | nM | 5.09 |
| CHEMBL5433156 | — | IC50 | = | 8068.0 | nM | 5.09 |
| CHEMBL5433711 | — | IC50 | = | 8237.0 | nM | 5.08 |
| CHEMBL5441124 | — | IC50 | = | 8275.0 | nM | 5.08 |
| CHEMBL5434414 | — | IC50 | = | 8578.0 | nM | 5.07 |
| CHEMBL5428502 | — | IC50 | = | 8491.0 | nM | 5.07 |
| CHEMBL5397012 | — | IC50 | = | 8608.0 | nM | 5.07 |
| CHEMBL5437898 | — | IC50 | = | 8534.0 | nM | 5.07 |
| CHEMBL5398897 | — | IC50 | = | 8534.0 | nM | 5.07 |
| CHEMBL5413820 | — | IC50 | = | 8687.0 | nM | 5.06 |
| CHEMBL5434519 | — | IC50 | = | 8747.0 | nM | 5.06 |
| CHEMBL5425117 | — | IC50 | = | 8793.0 | nM | 5.06 |
| CHEMBL5427329 | — | IC50 | = | 8848.0 | nM | 5.05 |
| CHEMBL5425539 | — | IC50 | = | 8873.0 | nM | 5.05 |
| CHEMBL5441132 | — | IC50 | = | 8907.0 | nM | 5.05 |
| CHEMBL5415366 | — | IC50 | = | 8889.0 | nM | 5.05 |
| CHEMBL5413463 | — | IC50 | = | 8818.0 | nM | 5.05 |
| CHEMBL5432496 | — | IC50 | = | 9074.0 | nM | 5.04 |
| CHEMBL5410090 | — | IC50 | = | 9062.0 | nM | 5.04 |
| CHEMBL5432722 | — | IC50 | = | 9186.0 | nM | 5.04 |
| CHEMBL5432224 | — | IC50 | = | 9172.0 | nM | 5.04 |
| CHEMBL5438169 | — | IC50 | = | 9067.0 | nM | 5.04 |
| CHEMBL5436859 | — | IC50 | = | 9357.0 | nM | 5.03 |
| CHEMBL5434537 | — | IC50 | = | 9875.0 | nM | 5.00 |
| CHEMBL5418432 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5425813 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5414065 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5407894 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5421438 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5430452 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5393904 | — | IC50 | > | 10000.0 | nM | - |