Assay Detail
Binding
CHEMBL5342184
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Agonist activity at TLR7 (unknown origin)
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Small-Molecule Modulators Targeting Toll-like Receptors for Potential Anticancer Therapeutics.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 18 | 6.50 | 8.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1082983 | — | — | 1 | 8.07 |
| CHEMBL5435648 | — | — | 1 | 7.80 |
| CHEMBL1086473 | — | — | 1 | 7.23 |
| CHEMBL5397718 | — | — | 1 | 7.07 |
| CHEMBL210884 | — | — | 1 | 6.85 |
| CHEMBL5268440 | — | — | 1 | 6.80 |
| CHEMBL5400758 | — | — | 1 | 6.72 |
| CHEMBL5276534 | — | — | 1 | 6.58 |
| CHEMBL5406749 | — | — | 1 | 6.57 |
| CHEMBL5430530 | — | — | 1 | 6.26 |
| CHEMBL5272163 | — | — | 1 | 6.07 |
| CHEMBL383322 | RESIQUIMOD | 2.0 | 1 | 5.82 |
| CHEMBL1085742 | — | — | 1 | 5.70 |
| CHEMBL1282 | IMIQUIMOD | 4.0 | 1 | 5.67 |
| CHEMBL5397171 | — | — | 1 | 4.36 |
| CHEMBL549344 | CPG-52852 | 2.0 | 1 | - |
| CHEMBL5418815 | — | — | 1 | - |
| CHEMBL5415035 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1082983 | — | EC50 | = | 8.58 | nM | 8.07 |
| CHEMBL5435648 | — | EC50 | = | 16.0 | nM | 7.80 |
| CHEMBL1086473 | — | EC50 | = | 59.1 | nM | 7.23 |
| CHEMBL5397718 | — | EC50 | = | 85.0 | nM | 7.07 |
| CHEMBL210884 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL5268440 | — | EC50 | = | 160.0 | nM | 6.80 |
| CHEMBL5400758 | — | EC50 | = | 190.0 | nM | 6.72 |
| CHEMBL5276534 | — | EC50 | = | 260.0 | nM | 6.58 |
| CHEMBL5406749 | — | EC50 | = | 270.0 | nM | 6.57 |
| CHEMBL5430530 | — | EC50 | = | 550.0 | nM | 6.26 |
| CHEMBL5272163 | — | EC50 | = | 860.0 | nM | 6.07 |
| CHEMBL383322 | RESIQUIMOD | EC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL1085742 | — | EC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL1282 | IMIQUIMOD | EC50 | = | 2120.0 | nM | 5.67 |
| CHEMBL5397171 | — | EC50 | = | 44000.0 | nM | 4.36 |
| CHEMBL549344 | CPG-52852 | EC50 | ~ | 3000.0 | nM | - |
| CHEMBL5418815 | — | EC50 | > | 100.0 | nM | - |
| CHEMBL5415035 | — | EC50 | > | 100.0 | nM | - |