Assay Detail
Functional
CHEMBL5343295
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Cytotoxicity against human Jurkat cells assessed as cell growth inhibition incubated for 48 hrs by MTT assay
43
Total Activities
43
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Jurkat |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Carbohydrate Strengthens the Immunotherapeutic Effect of Small-Molecule PD-L1 Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 43 | 4.73 | 5.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4089730 | — | — | 1 | 5.58 |
| CHEMBL5405710 | — | — | 1 | 5.55 |
| CHEMBL5425076 | — | — | 1 | 5.55 |
| CHEMBL5428162 | — | — | 1 | 5.39 |
| CHEMBL5431133 | — | — | 1 | 5.35 |
| CHEMBL5412775 | — | — | 1 | 5.27 |
| CHEMBL5394231 | — | — | 1 | 5.24 |
| CHEMBL5414674 | — | — | 1 | 5.21 |
| CHEMBL5434006 | — | — | 1 | 5.11 |
| CHEMBL5407204 | — | — | 1 | 5.06 |
| CHEMBL5425727 | — | — | 1 | 4.91 |
| CHEMBL5427156 | — | — | 1 | 4.83 |
| CHEMBL5423144 | — | — | 1 | 4.77 |
| CHEMBL5397889 | — | — | 1 | 4.75 |
| CHEMBL5432206 | — | — | 1 | 4.70 |
| CHEMBL5426080 | — | — | 1 | 4.61 |
| CHEMBL5406040 | — | — | 1 | 4.60 |
| CHEMBL5424608 | — | — | 1 | 4.59 |
| CHEMBL5408219 | — | — | 1 | 4.57 |
| CHEMBL5438626 | — | — | 1 | 4.56 |
| CHEMBL5397487 | — | — | 1 | 4.56 |
| CHEMBL5399366 | — | — | 1 | 4.51 |
| CHEMBL5424841 | — | — | 1 | 4.50 |
| CHEMBL5403695 | — | — | 1 | 4.46 |
| CHEMBL5400102 | — | — | 1 | 4.36 |
| CHEMBL5394157 | — | — | 1 | 4.36 |
| CHEMBL5408624 | — | — | 1 | 4.36 |
| CHEMBL5417900 | — | — | 1 | 4.34 |
| CHEMBL5422306 | — | — | 1 | 4.32 |
| CHEMBL5417055 | — | — | 1 | 4.31 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4089730 | — | IC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL5405710 | — | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL5425076 | — | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL5428162 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL5431133 | — | IC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL5412775 | — | IC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL5394231 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL5414674 | — | IC50 | = | 6200.0 | nM | 5.21 |
| CHEMBL5434006 | — | IC50 | = | 7800.0 | nM | 5.11 |
| CHEMBL5407204 | — | IC50 | = | 8800.0 | nM | 5.06 |
| CHEMBL5425727 | — | IC50 | = | 12400.0 | nM | 4.91 |
| CHEMBL5427156 | — | IC50 | = | 14900.0 | nM | 4.83 |
| CHEMBL5423144 | — | IC50 | = | 16900.0 | nM | 4.77 |
| CHEMBL5397889 | — | IC50 | = | 17900.0 | nM | 4.75 |
| CHEMBL5432206 | — | IC50 | = | 19800.0 | nM | 4.70 |
| CHEMBL5426080 | — | IC50 | = | 24500.0 | nM | 4.61 |
| CHEMBL5406040 | — | IC50 | = | 24900.0 | nM | 4.60 |
| CHEMBL5424608 | — | IC50 | = | 25500.0 | nM | 4.59 |
| CHEMBL5408219 | — | IC50 | = | 26700.0 | nM | 4.57 |
| CHEMBL5438626 | — | IC50 | = | 27600.0 | nM | 4.56 |
| CHEMBL5397487 | — | IC50 | = | 27300.0 | nM | 4.56 |
| CHEMBL5399366 | — | IC50 | = | 30800.0 | nM | 4.51 |
| CHEMBL5424841 | — | IC50 | = | 31300.0 | nM | 4.50 |
| CHEMBL5403695 | — | IC50 | = | 34300.0 | nM | 4.46 |
| CHEMBL5400102 | — | IC50 | = | 43400.0 | nM | 4.36 |
| CHEMBL5394157 | — | IC50 | = | 44000.0 | nM | 4.36 |
| CHEMBL5408624 | — | IC50 | = | 43500.0 | nM | 4.36 |
| CHEMBL5417900 | — | IC50 | = | 46000.0 | nM | 4.34 |
| CHEMBL5422306 | — | IC50 | = | 47500.0 | nM | 4.32 |
| CHEMBL5417055 | — | IC50 | = | 49200.0 | nM | 4.31 |
| CHEMBL5395778 | — | IC50 | = | 50500.0 | nM | 4.30 |
| CHEMBL5398822 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL5404220 | — | IC50 | = | 53100.0 | nM | 4.28 |
| CHEMBL5399839 | — | IC50 | = | 53900.0 | nM | 4.27 |
| CHEMBL5416072 | — | IC50 | = | 73900.0 | nM | 4.13 |
| CHEMBL5415266 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5426397 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5427820 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5428988 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5436798 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5399177 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5425908 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL5434059 | — | IC50 | > | 100000.0 | nM | - |