Assay Detail
Binding
CHEMBL5372966
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [K4]hPP from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQ
2
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
[<sup>3</sup>H]UR-JG102-A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y<sub>4</sub> Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.70 | 9.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | 2.0 | 2 | 9.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | Ki | = | 0.17 | nM | 9.77 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | Ki | = | 0.24 | nM | 9.62 |