Assay Detail
Binding
CHEMBL5372970
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]UR-KK200 from human Y4R expressed in CHO cells co-expressing Gqi5-mtAEQ
26
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
[<sup>3</sup>H]UR-JG102-A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y<sub>4</sub> Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 26 | 10.06 | 10.61 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5437701 | — | — | 2 | 10.61 |
| CHEMBL5422869 | — | — | 2 | 10.52 |
| CHEMBL5423253 | — | — | 2 | 10.50 |
| CHEMBL5435492 | — | — | 2 | 10.40 |
| CHEMBL5437695 | — | — | 2 | 10.18 |
| CHEMBL5421880 | — | — | 2 | 10.04 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | 2.0 | 2 | 10.02 |
| CHEMBL5396128 | — | — | 2 | 9.97 |
| CHEMBL5430318 | — | — | 2 | 9.96 |
| CHEMBL5398948 | — | — | 2 | 9.84 |
| CHEMBL5400627 | — | — | 2 | 9.80 |
| CHEMBL5428340 | — | — | 2 | 9.59 |
| CHEMBL5429140 | — | — | 2 | 9.49 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5437701 | — | Ki | = | 0.02455 | nM | 10.61 |
| CHEMBL5437701 | — | Ki | = | 0.026 | nM | 10.59 |
| CHEMBL5422869 | — | Ki | = | 0.0302 | nM | 10.52 |
| CHEMBL5422869 | — | Ki | = | 0.031 | nM | 10.51 |
| CHEMBL5423253 | — | Ki | = | 0.03162 | nM | 10.50 |
| CHEMBL5423253 | — | Ki | = | 0.036 | nM | 10.44 |
| CHEMBL5435492 | — | Ki | = | 0.03981 | nM | 10.40 |
| CHEMBL5435492 | — | Ki | = | 0.041 | nM | 10.39 |
| CHEMBL5437695 | — | Ki | = | 0.066 | nM | 10.18 |
| CHEMBL5437695 | — | Ki | = | 0.06607 | nM | 10.18 |
| CHEMBL5421880 | — | Ki | = | 0.0912 | nM | 10.04 |
| CHEMBL5421880 | — | Ki | = | 0.093 | nM | 10.03 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | Ki | = | 0.0955 | nM | 10.02 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | Ki | = | 0.1 | nM | 10.00 |
| CHEMBL5396128 | — | Ki | = | 0.1072 | nM | 9.97 |
| CHEMBL5396128 | — | Ki | = | 0.11 | nM | 9.96 |
| CHEMBL5430318 | — | Ki | = | 0.1096 | nM | 9.96 |
| CHEMBL5430318 | — | Ki | = | 0.12 | nM | 9.92 |
| CHEMBL5398948 | — | Ki | = | 0.1445 | nM | 9.84 |
| CHEMBL5398948 | — | Ki | = | 0.15 | nM | 9.82 |
| CHEMBL5400627 | — | Ki | = | 0.1585 | nM | 9.80 |
| CHEMBL5400627 | — | Ki | = | 0.17 | nM | 9.77 |
| CHEMBL5428340 | — | Ki | = | 0.257 | nM | 9.59 |
| CHEMBL5428340 | — | Ki | = | 0.26 | nM | 9.59 |
| CHEMBL5429140 | — | Ki | = | 0.3236 | nM | 9.49 |
| CHEMBL5429140 | — | Ki | = | 0.33 | nM | 9.48 |