Assay Detail
Functional
CHEMBL5372976
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human Y4R expressed in HEK293T cells by miniGsi assay
26
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293T |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
[<sup>3</sup>H]UR-JG102-A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y<sub>4</sub> Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 26 | 8.52 | 9.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5422869 | — | — | 2 | 9.05 |
| CHEMBL5437701 | — | — | 2 | 9.00 |
| CHEMBL5435492 | — | — | 2 | 8.96 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | 2.0 | 2 | 8.96 |
| CHEMBL5437695 | — | — | 2 | 8.80 |
| CHEMBL5421880 | — | — | 2 | 8.60 |
| CHEMBL5430318 | — | — | 2 | 8.59 |
| CHEMBL5398948 | — | — | 2 | 8.42 |
| CHEMBL5429140 | — | — | 2 | 8.33 |
| CHEMBL5423253 | — | — | 2 | 8.29 |
| CHEMBL5396128 | — | — | 2 | 8.09 |
| CHEMBL5400627 | — | — | 2 | 8.00 |
| CHEMBL5428340 | — | — | 2 | 7.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5422869 | — | EC50 | = | 0.89 | nM | 9.05 |
| CHEMBL5422869 | — | EC50 | = | 0.8913 | nM | 9.05 |
| CHEMBL5437701 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL5437701 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL5435492 | — | EC50 | = | 1.096 | nM | 8.96 |
| CHEMBL5435492 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | EC50 | = | 1.148 | nM | 8.94 |
| CHEMBL5437695 | — | EC50 | = | 1.6 | nM | 8.80 |
| CHEMBL5437695 | — | EC50 | = | 1.622 | nM | 8.79 |
| CHEMBL5421880 | — | EC50 | = | 2.512 | nM | 8.60 |
| CHEMBL5421880 | — | EC50 | = | 2.5 | nM | 8.60 |
| CHEMBL5430318 | — | EC50 | = | 2.6 | nM | 8.59 |
| CHEMBL5430318 | — | EC50 | = | 2.63 | nM | 8.58 |
| CHEMBL5398948 | — | EC50 | = | 3.8 | nM | 8.42 |
| CHEMBL5398948 | — | EC50 | = | 3.802 | nM | 8.42 |
| CHEMBL5429140 | — | EC50 | = | 4.7 | nM | 8.33 |
| CHEMBL5429140 | — | EC50 | = | 4.677 | nM | 8.33 |
| CHEMBL5423253 | — | EC50 | = | 5.129 | nM | 8.29 |
| CHEMBL5423253 | — | EC50 | = | 5.1 | nM | 8.29 |
| CHEMBL5396128 | — | EC50 | = | 8.1 | nM | 8.09 |
| CHEMBL5396128 | — | EC50 | = | 8.128 | nM | 8.09 |
| CHEMBL5400627 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL5400627 | — | EC50 | = | 10.47 | nM | 7.98 |
| CHEMBL5428340 | — | EC50 | = | 19.0 | nM | 7.72 |
| CHEMBL5428340 | — | EC50 | = | 19.95 | nM | 7.70 |