Assay Detail
Functional
CHEMBL5372977
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Agonist activity at human Y4R expressed in HEK293T cells incubated for 60 mins by cAMP CAMYEN assay
16
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293T |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
[<sup>3</sup>H]UR-JG102-A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y<sub>4</sub> Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 16 | 9.83 | 10.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5437695 | — | — | 2 | 10.30 |
| CHEMBL5430318 | — | — | 2 | 10.00 |
| CHEMBL5398948 | — | — | 2 | 9.90 |
| CHEMBL5423253 | — | — | 2 | 9.90 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | 2.0 | 2 | 9.85 |
| CHEMBL4873376 | — | — | 2 | 9.79 |
| CHEMBL5396128 | — | — | 2 | 9.71 |
| CHEMBL5428340 | — | — | 2 | 9.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5437695 | — | EC50 | = | 0.05012 | nM | 10.30 |
| CHEMBL5437695 | — | EC50 | = | 0.063 | nM | 10.20 |
| CHEMBL5430318 | — | EC50 | = | 0.1 | nM | 10.00 |
| CHEMBL5430318 | — | EC50 | = | 0.11 | nM | 9.96 |
| CHEMBL5398948 | — | EC50 | = | 0.1259 | nM | 9.90 |
| CHEMBL5423253 | — | EC50 | = | 0.1259 | nM | 9.90 |
| CHEMBL5398948 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | EC50 | = | 0.1413 | nM | 9.85 |
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | EC50 | = | 0.15 | nM | 9.82 |
| CHEMBL4873376 | — | EC50 | = | 0.1622 | nM | 9.79 |
| CHEMBL5423253 | — | EC50 | = | 0.17 | nM | 9.77 |
| CHEMBL4873376 | — | EC50 | = | 0.17 | nM | 9.77 |
| CHEMBL5396128 | — | EC50 | = | 0.195 | nM | 9.71 |
| CHEMBL5396128 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL5428340 | — | EC50 | = | 0.3981 | nM | 9.40 |
| CHEMBL5428340 | — | EC50 | = | 0.41 | nM | 9.39 |