Assay Detail
Binding
CHEMBL5372999
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Binding affinity to human Y4R under hypotonic sodium free condition
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
[<sup>3</sup>H]UR-JG102-A Radiolabeled Cyclic Peptide with High Affinity and Excellent Selectivity for the Neuropeptide Y Y<sub>4</sub> Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.85 | 10.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | 2.0 | 1 | 10.64 |
| CHEMBL5411178 | — | — | 1 | 9.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4540843 | PANCREATIC POLYPEPTIDE | Ki | = | 0.023 | nM | 10.64 |
| CHEMBL5411178 | — | Ki | = | 0.87 | nM | 9.06 |