Assay Detail
Functional
CHEMBL5523932
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human T47D cells assessed as reduction in cell viability incubated for 72 hrs by CCK-8 assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | T47D |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Progress in the controllability technology of PROTAC.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.82 | 7.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4215078 | — | — | 1 | 7.89 |
| CHEMBL5289882 | — | — | 1 | 7.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4215078 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL5289882 | — | IC50 | = | 18.0 | nM | 7.75 |