Assay Detail
Functional
CHEMBL5524115
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Agonist activity at human FPR1 expressed in HL-60 cells assessed as increase in calcium mobilization by FLIPR analysis
12
Total Activities
12
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HL-60 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The formyl peptide receptors FPR1 and FPR2 as targets for inflammatory disorders: recent advances in the development of small-molecule agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 12 | 5.87 | 7.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5568107 | — | — | 1 | 7.64 |
| CHEMBL5563666 | — | — | 1 | 6.96 |
| CHEMBL5561947 | — | — | 1 | 6.55 |
| CHEMBL405908 | — | — | 1 | 6.52 |
| CHEMBL329650 | — | — | 1 | 6.24 |
| CHEMBL5568086 | — | — | 1 | 5.80 |
| CHEMBL5561891 | — | — | 1 | 5.48 |
| CHEMBL5562604 | — | — | 1 | 5.39 |
| CHEMBL4162930 | — | — | 1 | 5.28 |
| CHEMBL4173645 | — | — | 1 | 5.27 |
| CHEMBL5562581 | — | — | 1 | 4.70 |
| CHEMBL5563847 | — | — | 1 | 4.62 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5568107 | — | EC50 | = | 23.0 | nM | 7.64 |
| CHEMBL5563666 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL5561947 | — | EC50 | = | 280.0 | nM | 6.55 |
| CHEMBL405908 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL329650 | — | EC50 | = | 570.0 | nM | 6.24 |
| CHEMBL5568086 | — | EC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL5561891 | — | EC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL5562604 | — | EC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL4162930 | — | EC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL4173645 | — | EC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL5562581 | — | EC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL5563847 | — | EC50 | = | 24000.0 | nM | 4.62 |