Assay Detail
Functional
CHEMBL5524136
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Agonist activity at FPR2 (unknown origin) in HEK293 cells
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
The formyl peptide receptors FPR1 and FPR2 as targets for inflammatory disorders: recent advances in the development of small-molecule agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 17 | 8.12 | 10.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5567819 | — | — | 1 | 10.15 |
| CHEMBL5563146 | — | — | 1 | 9.52 |
| CHEMBL5561530 | — | — | 1 | 9.40 |
| CHEMBL5561111 | — | — | 1 | 9.15 |
| CHEMBL5561975 | — | — | 1 | 8.77 |
| CHEMBL5557151 | — | — | 1 | 8.70 |
| CHEMBL5542471 | — | — | 1 | 8.52 |
| CHEMBL5560784 | — | — | 1 | 8.40 |
| CHEMBL5563899 | — | — | 1 | 8.40 |
| CHEMBL5531970 | — | — | 1 | 8.40 |
| CHEMBL3915698 | — | — | 1 | 8.12 |
| CHEMBL4755656 | — | — | 1 | 8.00 |
| CHEMBL1370052 | — | — | 1 | 7.82 |
| CHEMBL1289381 | — | — | 1 | 7.00 |
| CHEMBL1289260 | — | — | 1 | 6.40 |
| CHEMBL1289811 | — | — | 1 | 5.68 |
| CHEMBL1290250 | — | — | 1 | 5.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5567819 | — | EC50 | = | 0.07 | nM | 10.15 |
| CHEMBL5563146 | — | EC50 | = | 0.3 | nM | 9.52 |
| CHEMBL5561530 | — | EC50 | = | 0.4 | nM | 9.40 |
| CHEMBL5561111 | — | EC50 | = | 0.7 | nM | 9.15 |
| CHEMBL5561975 | — | EC50 | = | 1.7 | nM | 8.77 |
| CHEMBL5557151 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5542471 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL5560784 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5563899 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5531970 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3915698 | — | EC50 | = | 7.6 | nM | 8.12 |
| CHEMBL4755656 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL1370052 | — | EC50 | = | 15.0 | nM | 7.82 |
| CHEMBL1289381 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1289260 | — | EC50 | = | 400.0 | nM | 6.40 |
| CHEMBL1289811 | — | EC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL1290250 | — | EC50 | = | 2600.0 | nM | 5.58 |