Assay Detail
Binding
CHEMBL5524642
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Inhibition of GOAT (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Modulators for palmitoylation of proteins and small molecules.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.60 | 7.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5566124 | — | — | 1 | 7.22 |
| CHEMBL5532041 | — | — | 1 | 6.77 |
| CHEMBL4556712 | — | — | 1 | 5.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5566124 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL5532041 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL4556712 | — | IC50 | = | 1500.0 | nM | 5.82 |