Assay Detail
Binding
CHEMBL5526175
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of 125I-Calcitonin from rat CTR expressed in Baby hamster kidney cell membrane incubated for 120 mins by SPA method
18
Total Activities
18
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Kidney |
| Cell Type | Baby hamster kidney cell |
| Subcellular | Membrane |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
NN1213 - A Potent, Long-Acting, and Selective Analog of Human Amylin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 18 | 7.47 | 10.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3989767 | CALCITONIN SALMON | 4.0 | 1 | 10.52 |
| CHEMBL2103758 | PRAMLINTIDE | 4.0 | 1 | 8.23 |
| CHEMBL5567107 | — | — | 1 | 8.22 |
| CHEMBL5568414 | — | — | 1 | 8.12 |
| CHEMBL5554990 | — | — | 1 | 7.77 |
| CHEMBL5566450 | — | — | 1 | 7.49 |
| CHEMBL5556440 | — | — | 1 | 7.30 |
| CHEMBL5560328 | — | — | 1 | 7.30 |
| CHEMBL5568431 | — | — | 1 | 7.29 |
| CHEMBL5561117 | — | — | 1 | 7.25 |
| CHEMBL5560524 | — | — | 1 | 7.15 |
| CHEMBL5566453 | — | — | 1 | 7.05 |
| CHEMBL5568545 | — | — | 1 | 7.02 |
| CHEMBL5567446 | — | — | 1 | 7.01 |
| CHEMBL5568471 | — | — | 1 | 6.98 |
| CHEMBL5567377 | — | — | 1 | 6.87 |
| CHEMBL5568143 | — | — | 1 | 6.46 |
| CHEMBL5565993 | — | — | 1 | 6.45 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3989767 | CALCITONIN SALMON | IC50 | = | 0.03 | nM | 10.52 |
| CHEMBL2103758 | PRAMLINTIDE | IC50 | = | 5.834 | nM | 8.23 |
| CHEMBL5567107 | — | IC50 | = | 5.976 | nM | 8.22 |
| CHEMBL5568414 | — | IC50 | = | 7.545 | nM | 8.12 |
| CHEMBL5554990 | — | IC50 | = | 17.11 | nM | 7.77 |
| CHEMBL5566450 | — | IC50 | = | 32.74 | nM | 7.49 |
| CHEMBL5556440 | — | IC50 | = | 50.05 | nM | 7.30 |
| CHEMBL5560328 | — | IC50 | = | 49.81 | nM | 7.30 |
| CHEMBL5568431 | — | IC50 | = | 51.41 | nM | 7.29 |
| CHEMBL5561117 | — | IC50 | = | 55.64 | nM | 7.25 |
| CHEMBL5560524 | — | IC50 | = | 71.02 | nM | 7.15 |
| CHEMBL5566453 | — | IC50 | = | 89.17 | nM | 7.05 |
| CHEMBL5568545 | — | IC50 | = | 96.44 | nM | 7.02 |
| CHEMBL5567446 | — | IC50 | = | 96.92 | nM | 7.01 |
| CHEMBL5568471 | — | IC50 | = | 105.57 | nM | 6.98 |
| CHEMBL5567377 | — | IC50 | = | 134.99 | nM | 6.87 |
| CHEMBL5568143 | — | IC50 | = | 349.7 | nM | 6.46 |
| CHEMBL5565993 | — | IC50 | = | 355.75 | nM | 6.45 |