Assay Detail
Toxicity
CHEMBL5578999
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Hemolytic activity against human RBC incubated for 1 hr by microplate reader analysis
24
Total Activities
24
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Toxicity |
| Organism | Homo sapiens |
| Cell Type | Erythrocyte |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Computational Design of Pore-Forming Peptides with Potent Antimicrobial and Anticancer Activities.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 24 | 5.17 | 6.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL174 | AMPICILLIN | 4.0 | 1 | 6.05 |
| CHEMBL5590171 | — | — | 1 | 5.16 |
| CHEMBL5592498 | — | — | 1 | 4.31 |
| CHEMBL5592838 | — | — | 1 | - |
| CHEMBL5590515 | — | — | 1 | - |
| CHEMBL5594404 | — | — | 1 | - |
| CHEMBL5590247 | — | — | 1 | - |
| CHEMBL5594680 | — | — | 1 | - |
| CHEMBL5591216 | — | — | 1 | - |
| CHEMBL5593137 | — | — | 1 | - |
| CHEMBL5595754 | — | — | 1 | - |
| CHEMBL5593337 | — | — | 1 | - |
| CHEMBL5595052 | — | — | 1 | - |
| CHEMBL5592285 | — | — | 1 | - |
| CHEMBL5594579 | — | — | 1 | - |
| CHEMBL5591279 | — | — | 1 | - |
| CHEMBL5593135 | — | — | 1 | - |
| CHEMBL5590497 | — | — | 1 | - |
| CHEMBL5584167 | — | — | 1 | - |
| CHEMBL5583887 | — | — | 1 | - |
| CHEMBL5590306 | — | — | 1 | - |
| CHEMBL5594932 | — | — | 1 | - |
| CHEMBL5592715 | — | — | 1 | - |
| CHEMBL5592279 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL174 | AMPICILLIN | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL5590171 | — | IC50 | = | 6900.0 | nM | 5.16 |
| CHEMBL5592498 | — | IC50 | = | 49000.0 | nM | 4.31 |
| CHEMBL5592838 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5590515 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5594404 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5590247 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5594680 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5591216 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5593137 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5595754 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5593337 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5595052 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5592285 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5594579 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5591279 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5593135 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5590497 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5584167 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5583887 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5590306 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5594932 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5592715 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL5592279 | — | IC50 | > | 50000.0 | nM | - |